SCHEMBL7207035

SCHEMBL7207035

COc1ccc(S(=O)(=O)C(C)C(C)C(=O)O)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP1 P03956 8/20 0.54
MMP13 P45452 5/20 0.54
MMP2 P08253 8/20 0.50
MMP3 P08254 7/20 0.50
MMP9 P14780 5/20 0.50
MMP8 P22894 3/20 0.50
MMP7 P09237 1/20 0.50
MMP12 P39900 1/20 0.50
MMP14 P50281 1/20 0.50
MMP16 P51512 1/20 0.50
PKM P14618 2/20 0.48
SLC1A3 P43003 1/20 0.48
SLC1A2 P43004 1/20 0.48
SLC1A1 P43005 1/20 0.48
HTT P42858 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
PDE4A P27815 4/20 0.47
PDE4B Q07343 4/20 0.47
PDE4C Q08493 4/20 0.47
PDE4D Q08499 4/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7352846 0.83 MMP13 (0.60) MMP1MMP13MMP2MMP3MMP9
SCHEMBL7207784 0.80 MMP2 (0.54) MMP1MMP13MMP2MMP3MMP9
SCHEMBL6929276 0.80 MMP1 (0.70) MMP1MMP13MMP2MMP3MMP9
SCHEMBL7212138 0.79 MMP13 (0.54) MMP1MMP13MMP2MMP3MMP9
SCHEMBL7415077 0.76 MMP9 (0.53) MMP1MMP13MMP2MMP3MMP9
SCHEMBL4195254 0.76 PKM (0.61) MMP1MMP13MMP2MMP9MMP8
SCHEMBL7207041 0.76 MMP1 (0.61) MMP1MMP13MMP2MMP3MMP9
SCHEMBL7378975 0.75 SLC1A3 (0.61) MMP1MMP13MMP2MMP3MMP9
SCHEMBL8861380 0.75 SLC1A3 (0.61) MMP1MMP13MMP2MMP3MMP9
SCHEMBL7207763 0.75 MMP1 (0.49) MMP1MMP13MMP2MMP3MMP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0939628-B1 THIOL SULFONE METALLOPROTEASE INHIBITORS MONSANTO CO (US) 2003-03-05 EP disclosed
US-6013649-A BOND DISORDERS; AUTOIMMUNE DISEASES; ANTITUMOR AGENTS MONSANTO COMPANY (US) 2000-01-11 US disclosed
EP-0939628-A4 THIOL SULFONE METALLOPROTEASE INHIBITORS MONSANTO CO (US) 1999-12-22 EP disclosed
EP-0939628-A1 THIOL SULFONE METALLOPROTEASE INHIBITORS MONSANTO COMPANY (US) 1999-09-08 EP disclosed
WO-1998003164-A1 THIOL SULFONE METALLOPROTEASE INHIBITORS MONSANTO COMPANY (US) 1998-01-29 WO disclosed