SCHEMBL7218561

SCHEMBL7218561

C=CCn1c(Nc2ccc(C(=O)O)cc2)nc(=O)c2ccccc21

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 5/20 0.47
KMT2A Q03164 5/20 0.47
NPC1 O15118 3/20 0.47
RAB9A P51151 2/20 0.47
RXFP1 Q9HBX9 1/20 0.44
ATM Q13315 1/20 0.43
PTGER4 P35408 2/20 0.42
CDH1 P12830 1/20 0.41
CTNNB1 P35222 1/20 0.41
TCF7L2 Q9NQB0 1/20 0.41
PDE4B Q07343 2/20 0.41
PDE4D Q08499 2/20 0.41
RXRA P19793 1/20 0.41
NR4A2 P43354 1/20 0.41
ABCC1 P33527 1/20 0.40
ABCG2 Q9UNQ0 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C19 P33261 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7224196 0.88 CDH1 (0.52) MEN1KMT2ANPC1RAB9ARXFP1
SCHEMBL7224206 0.84 DRD2 (0.50) RXFP1ATMPTGER4CYP1A2CYP2C19
SCHEMBL7222312 0.83 MEN1 (0.41) MEN1KMT2ANPC1RAB9ACDH1
SCHEMBL7218618 0.83 MEN1 (0.42) MEN1KMT2ANPC1RAB9AKDM4E
SCHEMBL7224007 0.80 EGFR (0.50) MEN1KMT2ANPC1RAB9AATM
SCHEMBL7224034 0.77 CYP1A2 (0.47) MEN1KMT2ANPC1RAB9ARXFP1
SCHEMBL11840495 0.77 ALDH1A1 (0.46) MEN1KMT2ANPC1RAB9ARXFP1
SCHEMBL7217250 0.72 L3MBTL1 (0.49) MEN1KMT2ANPC1RAB9AKDM4E
SCHEMBL2359465 0.72 CYP1A2 (0.68) MEN1KMT2ANPC1RAB9ARXFP1
SCHEMBL9374216 0.70 ALDH1A1 (0.46) MEN1KMT2ANPC1RXFP1ATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6525061-B1 Combinatorial libraries for drug discovery;4-((6-bromo-4-oxo-1,4-dihydroquinazolin-2-yl)amino)b enzoic acid, WYETH 2003-02-25 US claimed
US-6525061-B1 Combinatorial libraries for drug discovery;4-((6-bromo-4-oxo-1,4-dihydroquinazolin-2-yl)amino)b enzoic acid, WYETH 2003-02-25 US disclosed