SCHEMBL7224007

SCHEMBL7224007

Cn1c(Nc2ccc(C(=O)O)cc2)nc(=O)c2ccccc21

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 4/20 0.50
KDM4E B2RXH2 3/20 0.50
SRC P12931 3/20 0.50
ATM Q13315 1/20 0.50
HSD17B10 Q99714 1/20 0.49
MEN1 O00255 3/20 0.48
KMT2A Q03164 3/20 0.48
NPC1 O15118 2/20 0.48
MAPT P10636 2/20 0.48
RAB9A P51151 2/20 0.48
GAA P10253 1/20 0.48
HDAC6 Q9UBN7 1/20 0.48
ABCC1 P33527 1/20 0.46
ABCG2 Q9UNQ0 1/20 0.46
KDR P35968 1/20 0.46
TP53 P04637 1/20 0.46
HPGD P15428 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
SIRT5 Q9NXA8 1/20 0.45
GSK3A P49840 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13977074 0.87 KDM4E (0.57) KDM4EHSD17B10NPC1MAPTRAB9A
SCHEMBL7217219 0.86 L3MBTL1 (0.54) EGFRKDM4ESRCHSD17B10MEN1
SCHEMBL9910545 0.82 NPC1 (0.62) ATMHSD17B10MEN1KMT2ANPC1
SCHEMBL7224206 0.82 DRD2 (0.50) KDM4EATMMAPTHDAC6PTGER4
SCHEMBL7218561 0.80 MEN1 (0.47) EGFRKDM4EATMMEN1KMT2A
SCHEMBL9728470 0.77 RAB9A (0.68) KDM4EHSD17B10MEN1KMT2ANPC1
SCHEMBL9728272 0.74 RAB9A (0.56) KDM4EHSD17B10MEN1KMT2ANPC1
SCHEMBL7223862 0.72 KDM4E (0.46) EGFRKDM4ESRCHSD17B10KMT2A
SCHEMBL2724437 0.71 HSD17B10 (0.74) KDM4EATMHSD17B10KMT2ANPC1
SCHEMBL9729063 0.71 MAPK1 (0.57) KDM4EHSD17B10KMT2ANPC1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6525061-B1 Combinatorial libraries for drug discovery;4-((6-bromo-4-oxo-1,4-dihydroquinazolin-2-yl)amino)b enzoic acid, WYETH 2003-02-25 US claimed
US-6525061-B1 Combinatorial libraries for drug discovery;4-((6-bromo-4-oxo-1,4-dihydroquinazolin-2-yl)amino)b enzoic acid, WYETH 2003-02-25 US disclosed