SCHEMBL7223301

SCHEMBL7223301

CC(=O)c1ccc(Oc2ccc(C(=O)N[C@@H]3C[C@H]4CC[C@@H]3N4)s2)cc1

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.36
HPGD P15428 1/20 0.36
RAB9A P51151 1/20 0.36
ICAM1 P05362 1/20 0.33
SELE P16581 1/20 0.33
HTR3E A5X5Y0 1/20 0.33
HTR3B O95264 1/20 0.33
HTR3A P46098 1/20 0.33
HTR3D Q70Z44 1/20 0.33
HTR3C Q8WXA8 1/20 0.33
MMP2 P08253 1/20 0.32
MMP7 P09237 1/20 0.32
MMP9 P14780 1/20 0.32
MMP13 P45452 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
SLC6A4 P31645 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7116899 0.92 MMP2 (0.36) MAPTHTR3EHTR3BHTR3AHTR3D
SCHEMBL7224931 0.90 F2 (0.37) MMP2MMP7MMP9MMP13KMT2A
SCHEMBL7225149 0.90 HTR4 (0.37) MAPTHPGDRAB9ASLC6A4
SCHEMBL7229845 0.90 SLC6A3 (0.42) RAB9AMMP13SLC6A4
SCHEMBL7233323 0.89 ESR1 (0.37) HPGDSLC6A4
SCHEMBL7232389 0.88 NPC1 (0.36) RAB9AHTR3EHTR3BHTR3AHTR3D
SCHEMBL7231735 0.88 MMP2 (0.36) MAPTICAM1SELEMMP2MMP7
SCHEMBL7225066 0.88 SLC6A4 (0.41) KMT2ASLC6A4
SCHEMBL7232095 0.88 CHRNA7 (0.34) HPGDSLC6A4
SCHEMBL7225381 0.87 HTR3E (0.37) HTR3EHTR3BHTR3AHTR3DHTR3C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US claimed
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US disclosed