SCHEMBL7225301

SCHEMBL7225301

O=C(N[C@@H]1C[C@H]2CC[C@@H]1N2)c1ccc(Oc2cncc(Cl)c2)s1

nearest known ligand 0.39

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CCNC P24863 1/20 0.37
CDK8 P49336 1/20 0.37
ADRB1 P08588 1/20 0.34
ADRB3 P13945 1/20 0.34
CHRNB2 P17787 4/20 0.33
CHRNA4 P43681 4/20 0.33
SLC6A3 Q01959 3/20 0.33
SLC6A4 P31645 2/20 0.33
PTGER4 P35408 1/20 0.32
F10 P00742 1/20 0.32
SMYD3 Q9H7B4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7225045 0.87 SLC6A3 (0.41) ADRB1ADRB3SLC6A3SLC6A4
SCHEMBL7225066 0.86 SLC6A4 (0.41) CCNCCDK8ADRB1ADRB3CHRNB2
SCHEMBL7225892 0.85 CHRNB2 (0.39) CHRNB2CHRNA4
SCHEMBL7225557 0.85 SLC8A1 (0.37) CHRNB2CHRNA4
SCHEMBL7231264 0.84 CYP1A2 (0.32) SLC6A3SLC6A4F10
SCHEMBL7223948 0.83 TAS1R3 (0.36) CHRNB2CHRNA4SLC6A3SLC6A4
SCHEMBL7124913 0.82 MMP2 (0.39) PTGER4SMYD3
SCHEMBL7223860 0.82 SLC6A4 (0.36) CCNCCDK8CHRNB2CHRNA4SLC6A3
SCHEMBL7225381 0.82 HTR3E (0.37) SLC6A3SLC6A4
SCHEMBL7234416 0.82 F10 (0.37) SLC6A3SLC6A4F10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US claimed
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US disclosed