Water

Water

SCHEMBL7227622

NC(CC(=O)O)C(N)CC(=O)O.O.O

nearest known ligand 0.47

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABCC9ABL1ACEACHEACVR1ADORA1ADORA2AADORA2BADORA3ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3AGTR1ALOX5ATP4AATP4BBCRBTKCACNA1ACACNA1BCACNA1CCACNA1DCACNA1ECACNA1FCACNA1GCACNA1HCACNA1ICACNA1SCACNA2D1CACNA2D2CACNA2D3CACNA2D4CACNB1CACNB2CACNB3CACNB4CACNG1CACNG2CACNG3CACNG4CACNG5CACNG6CACNG7CACNG8CALCRLCFBCHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNB1CHRNDCHRNECHRNGCRBNCUL4ACXCR1CXCR2DDB1DDCDHFRDPP4DRD2DRD3DRD4EGFRERBB2ERBB4ESR1ESR2FDPSFKBP1AFLT1FLT3FLT4GARTGHSRGRIA1GRIA2GRIA3GRIA4GRIK1GRIK2GRIK3GRIK4GRIK5GRIN2AGSK3AGSK3BHDAC1HDAC10HDAC11HDAC2HDAC3HDAC4HDAC5HDAC6HDAC7HDAC8HDAC9HRH1HTR1AHTR1BHTR1DHTR1EHTR1FHTR2AHTR2BHTR2CHTR3AHTR3BHTR3CHTR3DHTR3EHTR4HTR5AHTR6HTR7IDH1IDH2IMPA1ITGA2BITGB3JAK1JAK2JAK3KCNJ11KCNK3KCNK9KDRKITMEN1METMMP1MMP13MMP7MMP8NANOD2NS5bODC1OPG057OPRD1OPRK1OPRM1PPARP1PARP2PDE3APDE3BPDE4APDE4BPDE4CPDE4DPDGFRBPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PKLRPPARDPPATPTGS1PTGS2RBX1ROCK1ROCK2RRM1RRM2RRM2BSCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASCNN1ASCNN1BSCNN1GSIGMAR1SLC10A2SLC5A2SLC6A2SLC6A3SLC6A4SLC9A3SYKTACR1THRATHRBTOP1TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYK2TYMSVDRampCblablaT-3blaT-4blaT-5blaT-6blaUOE-1dacAdacBdacCfolAfolPftsIgyrAgyrBileSmecAmrcAmrcBmrdAparCparEpbp2pbp4pbpApbpFrplArplBrplCrplDrplErplFrplIrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmE2rpmFrpmGrpmG1rpmG2rpmG3rpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUthyAykgMykgO

The experimentally established mechanism targets of Water. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIK1 known ✓ P39086 1/20 0.38
GRIA1 known ✓ P42261 1/20 0.38
GRIA2 known ✓ P42262 1/20 0.38
GRIA3 known ✓ P42263 1/20 0.38
GRIA4 known ✓ P48058 1/20 0.38
GRIN2A known ✓ Q12879 1/20 0.38
GRIK2 known ✓ Q13002 1/20 0.38
GRIK3 known ✓ Q13003 1/20 0.38
GRIK5 known ✓ Q16478 1/20 0.38
CACNA2D1 known ✓ P54289 2/20 0.37
CACNB3 known ✓ P54284 1/20 0.37
CACNA1C known ✓ Q13936 1/20 0.37
ADRA1A known ✓ P35348 1/20 0.37
HTR2B known ✓ P41595 1/20 0.37
CACNA2D2 known ✓ Q9NY47 1/20 0.37
SLC22A6 Q4U2R8 1/20 0.47
GABRR1 P24046 2/20 0.46
LMNA P02545 1/20 0.46
TDP1 Q9NUW8 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2491274 0.97 SLC22A6 (0.50) SLC22A6GABRR1LMNATDP1SMN1; SMN2
SCHEMBL10657294 0.85 SLC22A6 (0.41) SLC22A6GABRR1LMNATDP1SMN1; SMN2
SCHEMBL10657150 0.85 SLC22A6 (0.41) SLC22A6GABRR1LMNATDP1SMN1; SMN2
SCHEMBL740306 0.84
SCHEMBL10655250 0.83 MAPT (0.39) SLC22A6GABRR1LMNATDP1SMN1; SMN2
SCHEMBL18980805 0.83 MAPT (0.39) SLC22A6GABRR1LMNATDP1SMN1; SMN2
SCHEMBL10653694 0.83 MAPT (0.39) SLC22A6GABRR1LMNATDP1SMN1; SMN2
SCHEMBL23225427 0.81
SCHEMBL17234502 0.79
SCHEMBL10657948 0.79

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6627580-B2 Conjugated imines that are selectivite for tri-valent manganese ions; used for the treatment of manganese deficiency in plant cultivation AKZO NOBEL N.V. (NL) 2003-09-30 US disclosed
US-20020156308-A1 Conjugated imines that are selectivite for tri-valent manganese ions; used for the treatment of manganese deficiency in plant cultivation HAKANSON CHRISTER L (SE) 2002-10-24 US disclosed
US-6458980-B1 MANGANIC CHELATES OF THE CHELATING AGENTS AND SALTS WITH PERMANGANATE OR MANGANESE DIOXIDE CHELATING AGENTS (CHELANTS) OF THE GENERAL STRUCTURE: DEFICIENCY IN PLANT CULTIVATION. AKZO NOBEL NV (NL) 2002-10-01 US disclosed
EP-0998450-A1 CHELATING AGENTS AND THEIR MANGANIC CHELATES Akzo Nobel N.V. (NL) 2000-05-10 EP disclosed
WO-1999002487-A1 CHELATING AGENTS AND THEIR MANGANIC CHELATES AKZO NOBEL N.V. (NL) 1999-01-21 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020156308-A1 Conjugated imines that are selectivite for tri-valent manganese ions; used for the treatment of manganese deficiency in plant cultivation MT-CO2, ZC3HAV1, MT-CO1 GRIK1 1688/4885GRIA1 863/4885GRIA2 644/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.