SCHEMBL7234263

SCHEMBL7234263

CN(C)c1ccc(CN2CCCN(c3ncccc3C(=O)O)CC2)cc1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.49
ALDH1A1 P00352 3/20 0.48
HTR3E A5X5Y0 2/20 0.44
HTR3B O95264 2/20 0.44
HTR3A P46098 2/20 0.44
HTR3D Q70Z44 2/20 0.44
HTR3C Q8WXA8 2/20 0.44
HTR1A P08908 1/20 0.44
HTR2C P28335 1/20 0.44
HSD11B1 P28845 1/20 0.44
KDM4E B2RXH2 1/20 0.43
TSHR P16473 2/20 0.43
HSD17B10 Q99714 1/20 0.43
HSP90AB1 P08238 1/20 0.41
CCR2 P41597 1/20 0.41
CHIA Q9BZP6 1/20 0.41
HTT P42858 1/20 0.41
ACKR3 P25106 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7239131 0.87 KDM4E (0.48) ALDH1A1HSD11B1KDM4ECHIAHTT
SCHEMBL7238619 0.85 L3MBTL1 (0.54) KMT2AHSD17B10
SCHEMBL7235226 0.83 HTR3E (0.61) KMT2AALDH1A1HTR3EHTR3BHTR3A
SCHEMBL7242879 0.82 CAPN1 (0.47) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL7235461 0.82 CAPN1 (0.47) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL7239796 0.81 SIGMAR1 (0.54) KMT2AALDH1A1HSD17B10
SCHEMBL7238307 0.79 TSHR (0.48) ALDH1A1HTR3EHTR3BHTR3AHTR3D
SCHEMBL2222747 0.78 HTR3E (0.53) KMT2AALDH1A1HTR3EHTR3BHTR3A
SCHEMBL7235600 0.78 ALDH1A1 (0.53) KMT2AALDH1A1TSHR
SCHEMBL15294735 0.78 KMT2A (0.70) KMT2AALDH1A1KDM4ETSHRHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6562827-B1 For the treatment of diseases in which increased calpain activity occurs such as neurodegenerative diseases or neuronal damage are caused by ischemia, trauma or mass hemorrhages ABBOTT LABORATORIES 2003-05-13 US disclosed