SCHEMBL7269669

SCHEMBL7269669

c1ccc(OCC2(COc3ccccc3)CO2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNA3 P22001 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
TAAR1 Q96RJ0 1/20 0.40
ALDH1A1 P00352 1/20 0.40
RECQL P46063 1/20 0.40
ALOX15 P16050 1/20 0.39
HTR1A P08908 1/20 0.38
ADRA1A P35348 1/20 0.38
LTA4H P09960 1/20 0.38
MAOB P27338 2/20 0.37
MAOA P21397 1/20 0.37
HDAC3 O15379 1/20 0.36
HDAC4 P56524 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC7 Q8WUI4 1/20 0.36
HDAC2 Q92769 1/20 0.36
HDAC10 Q969S8 1/20 0.36
HDAC11 Q96DB2 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4451944 0.88 LTA4H (0.41) KCNA3TDP1TAAR1ALDH1A1RECQL
SCHEMBL27760167 0.88 TAAR1 (0.44) KCNA3TDP1TAAR1ALDH1A1RECQL
SCHEMBL476346 0.87 TDP1 (0.38) KCNA3TDP1TAAR1ALDH1A1RECQL
SCHEMBL7218155 0.84 THRB (0.38) KCNA3TDP1TAAR1ALDH1A1RECQL
SCHEMBL246844 0.82 TDP1 (0.54) TDP1ALDH1A1HTR1AADRA1A
SCHEMBL667989 0.79 KCNA3 (0.41) KCNA3TDP1TAAR1ALDH1A1RECQL
SCHEMBL11013902 0.79 ALDH1A1 (0.42) KCNA3TDP1TAAR1ALDH1A1RECQL
SCHEMBL19091769 0.79 KCNA3 (0.41) KCNA3TDP1TAAR1ALDH1A1RECQL
SCHEMBL11264607 0.78 HTR1A (0.48) KCNA3TDP1TAAR1ALDH1A1RECQL
SCHEMBL11399029 0.77 LTA4H (0.39) KCNA3TDP1HTR1ALTA4HMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0839798-A2 Intermediates for preparating non-peptide retroviral protease inhibitors ABBOTT LABORATORIES (US) 1998-05-06 EP disclosed
US-5670675-A Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1997-09-23 US disclosed
US-5545750-A TREATING HUMAN IMMUNODEFICIENCY VIRUS ABBOTT LABORATORIES (US) 1996-08-13 US disclosed
US-5142056-A Human immunodeficiency virus protease inhibitor ABBOTT LABORATORIES (US) 1992-08-25 US disclosed
EP-0402646-A1 Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1990-12-19 EP disclosed