SCHEMBL7272984

SCHEMBL7272984

C=CC[C@@H]1C[C@@H](CC(N)=O)N(CCCc2ccccc2)C1=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNB4 P30926 1/20 0.39
CHRNA3 P32297 1/20 0.39
OPRM1 P35372 2/20 0.38
OPRD1 P41143 2/20 0.38
FAAH O00519 5/20 0.37
ALDH1A1 P00352 4/20 0.36
TSHR P16473 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
PARP1 P09874 1/20 0.36
PARP2 Q9UGN5 1/20 0.36
SIGMAR1 Q99720 2/20 0.36
ELANE P08246 1/20 0.35
MGLL Q99685 2/20 0.35
MEN1 O00255 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7275324 0.86 CHRNB4 (0.39) CHRNB4CHRNA3FAAHALDH1A1NPC1
SCHEMBL7275478 0.86 CHRNB4 (0.39) CHRNB4CHRNA3FAAHALDH1A1NPC1
SCHEMBL7274379 0.86 FAAH (0.39) CHRNB4CHRNA3OPRM1FAAHALDH1A1
SCHEMBL7273681 0.86 ALDH1A1 (0.44) OPRM1OPRD1ALDH1A1TSHRSMN1; SMN2
SCHEMBL7283442 0.83 GAA (0.39) CHRNB4CHRNA3FAAHTSHRNPC1
SCHEMBL7274559 0.82 OPRM1 (0.39) OPRM1SIGMAR1KCNH2
SCHEMBL7276423 0.81 FAAH (0.37) CHRNB4CHRNA3OPRM1FAAHALDH1A1
SCHEMBL7273909 0.80 TDP1 (0.44) ALDH1A1TSHRSMN1; SMN2RAB9AKMT2A
SCHEMBL7272672 0.79 ALDH1A1 (0.39) OPRM1FAAHALDH1A1SMN1; SMN2SIGMAR1
SCHEMBL7274062 0.79 ALDH1A1 (0.39) OPRM1ALDH1A1SMN1; SMN2SIGMAR1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0483667-B1 Cyclic imino derivatives, process for their preparation and drugs containing them THOMAE GMBH DR K (DE) 1998-02-04 EP disclosed
US-5591769-A PYRROLIDINE DERIVATIVES; ANTICOAGULANTS KARL THOMAE GMBH (DE) 1997-01-07 US disclosed
US-5541343-A ANTIAGGLOMERANTS FOR CELLS OR ANTICOAGULANTS KARL THOMAE GMBH (DE) 1996-07-30 US disclosed
EP-0483667-A2 Cyclic imino derivatives, process for their preparation and drugs containing them Dr. Karl Thomae GmbH (DE) 1992-05-06 EP disclosed