SCHEMBL7274430

SCHEMBL7274430

NC1Cc2ccc(CC(=O)NC[C@@H]3C[C@@H](CC(=O)O)C(=O)N3CCCc3ccccc3)cc2C1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 3/20 0.35
ITGB3 P05106 3/20 0.34
ITGA2B P08514 3/20 0.34
GAA P10253 1/20 0.34
HPGD P15428 1/20 0.34
ALDH1A1 P00352 2/20 0.33
ITGB1 P05556 1/20 0.33
ITGA5 P08648 1/20 0.33
TSHR P16473 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
NAMPT P43490 2/20 0.33
TRPV1 Q8NER1 2/20 0.33
LTA4H P09960 1/20 0.33
MEN1 O00255 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7276603 0.92 TBXA2R (0.35) MTNR1AITGB3ITGA2BGAAHPGD
SCHEMBL7284272 0.89 ITGB3 (0.37) MTNR1AITGB3ITGA2BGAAHPGD
SCHEMBL7274663 0.87 ITGB3 (0.40) MTNR1AITGB3ITGA2BALDH1A1TSHR
SCHEMBL7336889 0.85 SIGMAR1 (0.37) MTNR1AITGB3ITGA2BKMT2A
SCHEMBL7274241 0.85 SIGMAR1 (0.39) MTNR1AITGB3ITGA2BNAMPTLTA4H
Water SCHEMBL7275459 0.82 PNMT (0.41) ALDH1A1TSHRSMN1; SMN2TBXA2R
SCHEMBL7274427 0.81 ITGB3 (0.35) ITGB3ITGA2BALDH1A1TSHRSMN1; SMN2
SCHEMBL7275950 0.80 LTA4H (0.43) MTNR1AALDH1A1TSHRSMN1; SMN2LTA4H
SCHEMBL7280208 0.80 LTA4H (0.43) MTNR1AALDH1A1TSHRSMN1; SMN2LTA4H
SCHEMBL7282210 0.80 SIGMAR1 (0.44) MTNR1AHPGDALDH1A1TSHRSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0483667-B1 Cyclic imino derivatives, process for their preparation and drugs containing them THOMAE GMBH DR K (DE) 1998-02-04 EP disclosed
US-5591769-A PYRROLIDINE DERIVATIVES; ANTICOAGULANTS KARL THOMAE GMBH (DE) 1997-01-07 US disclosed
US-5541343-A ANTIAGGLOMERANTS FOR CELLS OR ANTICOAGULANTS KARL THOMAE GMBH (DE) 1996-07-30 US disclosed
EP-0483667-A2 Cyclic imino derivatives, process for their preparation and drugs containing them Dr. Karl Thomae GmbH (DE) 1992-05-06 EP disclosed