SCHEMBL7275946

SCHEMBL7275946

CC(C)[C@H](NC(=O)OCc1ccccc1)C(=O)OC(Cc1ccccc1)C1OC(C)(C)OC1C(Cc1ccccc1)OC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)C

nearest known ligand 0.52

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 1/20 0.47
CASP3 P42574 1/20 0.47
CASP7 P55210 1/20 0.47
CASP6 P55212 1/20 0.47
CASP8 Q14790 1/20 0.47
CTSS P25774 3/20 0.47
CTSL P07711 2/20 0.47
CTSB P07858 2/20 0.47
CTSK P43235 2/20 0.47
CAPN1 P07384 2/20 0.46
CCR1 P32246 2/20 0.46
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
CTSD P07339 1/20 0.45
ECE1 P42892 2/20 0.45
ATM Q13315 1/20 0.45
MME P08473 1/20 0.45
CTRB1 P17538 2/20 0.45
TRPM8 Q7Z2W7 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9709105 0.78 PYGL (0.49)
SCHEMBL7277492 0.77 CTSD (0.55) CASP1CASP3CASP7CASP6CASP8
SCHEMBL3733900 0.76 CTSL (0.57) CASP1CASP3CASP7CASP6CASP8
SCHEMBL3725467 0.76 CTSL (0.57) CASP1CASP3CASP7CASP6CASP8
SCHEMBL28949078 0.76 CTSL (0.57) CASP1CASP3CASP7CASP6CASP8
SCHEMBL16869639 0.76 CASP1 (0.46) CASP1CASP3CASP7CASP6CASP8
SCHEMBL10535596 0.75 TRPM8 (0.62) CASP1CASP3CASP7CASP6CASP8
SCHEMBL1908598 0.75 CTSK (0.62) CASP1CASP3CASP7CASP6CASP8
SCHEMBL10535601 0.75 TRPM8 (0.62) CASP1CASP3CASP7CASP6CASP8
SCHEMBL28892051 0.75 TRPM8 (0.62) CASP1CASP3CASP7CASP6CASP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0839798-A2 Intermediates for preparating non-peptide retroviral protease inhibitors ABBOTT LABORATORIES (US) 1998-05-06 EP disclosed
US-5670675-A Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1997-09-23 US disclosed
US-5545750-A TREATING HUMAN IMMUNODEFICIENCY VIRUS ABBOTT LABORATORIES (US) 1996-08-13 US disclosed
EP-0402646-A1 Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1990-12-19 EP disclosed