SCHEMBL7280264

SCHEMBL7280264

C=CC[C@@H]1C[C@@H](CNC(=O)c2cccc(C#N)c2)N(CCCc2ccccc2)C1=O

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 2/20 0.43
HTR1A P08908 2/20 0.41
NAMPT P43490 3/20 0.40
DRD3 P35462 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
DRD4 P21917 1/20 0.38
CHRM3 P20309 1/20 0.38
MAOA P21397 1/20 0.38
MCHR1 Q99705 1/20 0.37
GPR139 Q6DWJ6 1/20 0.37
CCR5 P51681 1/20 0.37
ROCK2 O75116 1/20 0.36
CTSL P07711 1/20 0.36
CTSB P07858 1/20 0.36
CTSK P43235 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7275535 0.91 CCR3 (0.43) DRD2HTR1ANAMPTHDAC8HDAC6
SCHEMBL7281678 0.89 HTR1A (0.42) DRD2HTR1ANAMPTDRD3HDAC8
SCHEMBL7284443 0.88 DRD2 (0.38) DRD2NAMPTDRD3HDAC8HDAC6
SCHEMBL7284718 0.86 HTR1A (0.42) DRD2HTR1ANAMPTDRD3DRD4
SCHEMBL7280648 0.83 HTR1A (0.41) DRD2HTR1ADRD4
SCHEMBL7280539 0.81 SIGMAR1 (0.44) DRD2HTR1ANAMPTDRD3MAOA
SCHEMBL7274964 0.79 CCR3 (0.44) HTR1ANAMPTHDAC6DRD4MAOA
Methyl Alcohol SCHEMBL8879759 0.79 HTR1A (0.40) DRD2HTR1ANAMPTDRD3HDAC6
SCHEMBL7278834 0.78 HTR1A (0.39) HTR1ANAMPTHDAC6CHRM3
SCHEMBL7273369 0.78 MAOA (0.38) DRD2HTR1ANAMPTDRD3MAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0483667-B1 Cyclic imino derivatives, process for their preparation and drugs containing them THOMAE GMBH DR K (DE) 1998-02-04 EP disclosed
US-5591769-A PYRROLIDINE DERIVATIVES; ANTICOAGULANTS KARL THOMAE GMBH (DE) 1997-01-07 US disclosed
US-5541343-A ANTIAGGLOMERANTS FOR CELLS OR ANTICOAGULANTS KARL THOMAE GMBH (DE) 1996-07-30 US disclosed
EP-0483667-A2 Cyclic imino derivatives, process for their preparation and drugs containing them Dr. Karl Thomae GmbH (DE) 1992-05-06 EP disclosed