SCHEMBL7304233

SCHEMBL7304233

COc1ccc(C2=CCN(CCCNC(=O)N3CCCC3=O)CC2)cc1OC

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.49
POLB P06746 1/20 0.43
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
DRD3 P35462 1/20 0.42
L3MBTL1 Q9Y468 2/20 0.41
QDPR P09417 2/20 0.41
ALDH1A1 P00352 2/20 0.41
TMEM97 Q5BJF2 1/20 0.41
TLR9 Q9NR96 1/20 0.40
TLR8 Q9NR97 1/20 0.40
TLR7 Q9NYK1 1/20 0.40
HPGD P15428 1/20 0.40
HSD17B10 Q99714 1/20 0.40
HTR7 P34969 1/20 0.40
KMT2A Q03164 1/20 0.40
PDE4B Q07343 1/20 0.39
HTR1A P08908 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7299309 0.89 SIGMAR1 (0.49) SIGMAR1CYP2D6CYP2C9DRD3ALDH1A1
SCHEMBL7297853 0.84 SIGMAR1 (0.48) SIGMAR1ALDH1A1HTR7KMT2AHTR1A
SCHEMBL7333358 0.84 HTR1A (0.48) SIGMAR1POLBALDH1A1HPGDHSD17B10
SCHEMBL9372501 0.84 SIGMAR1 (0.52) SIGMAR1HTR1A
SCHEMBL7335487 0.81 SIGMAR1 (0.47) SIGMAR1DRD3HSD17B10HTR7KMT2A
Fumaric Acid SCHEMBL9375443 0.79 SIGMAR1 (0.46) SIGMAR1DRD3HSD17B10HTR7KMT2A
Maleic Acid SCHEMBL9375437 0.79 SIGMAR1 (0.46) SIGMAR1DRD3HSD17B10HTR7KMT2A
SCHEMBL9735887 0.79 PARP1 (0.45) SIGMAR1DRD3HTR7HTR1A
SCHEMBL9371817 0.78 HTR1A (0.56) SIGMAR1HTR1A
SCHEMBL9464104 0.68 RAB9A (0.50) CYP2D6CYP2C9ALDH1A1HPGDKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5149817-A Psychotropic agents SHIONOGI & CO., LTD. (JP) 1992-09-22 US disclosed
EP-0445701-A1 Novel tetrahydropyridine derivatives SHIONOGI SEIYAKU KABUSHIKI KAISHA trading under the name of SHIONOGI & CO. LTD. (JP) 1991-09-11 EP disclosed