SCHEMBL7305458

SCHEMBL7305458

CSCC[C@H](NCC(c1ccccc1)c1ccccc1)C(=O)NC(=O)OC(C)(C)C

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSK P43235 4/20 0.46
CTSS P25774 2/20 0.46
KLK5 Q9Y337 1/20 0.42
KLK7 P49862 1/20 0.42
CA2 P00918 1/20 0.42
ALDH1A1 P00352 2/20 0.41
MEN1 O00255 1/20 0.41
LMNA P02545 1/20 0.41
TSHR P16473 1/20 0.41
KMT2A Q03164 1/20 0.41
HSD17B10 Q99714 1/20 0.41
FNTA P49354 1/20 0.41
FNTB P49356 1/20 0.41
PGGT1B P53609 1/20 0.41
BACE1 P56817 3/20 0.40
KDM4E B2RXH2 2/20 0.40
MAPT P10636 1/20 0.40
EPHX2 P34913 1/20 0.40
PPARG P37231 1/20 0.39
PPARA Q07869 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7317918 0.93 CTSK (0.46) CTSKCTSSKLK5KLK7CA2
SCHEMBL7317017 0.85 CTSK (0.47) CTSKCTSSKLK5KLK7CA2
SCHEMBL7307839 0.85 ANPEP (0.49) CTSKCTSSKLK5KLK7ALDH1A1
SCHEMBL7311059 0.84 CTSK (0.47) CTSKCTSSKLK5KLK7CA2
SCHEMBL7316663 0.84 CA2 (0.53) CTSKCTSSKLK5KLK7CA2
SCHEMBL7301520 0.82 CTSK (0.44) CTSKCTSSALDH1A1MEN1KMT2A
SCHEMBL7313561 0.79 CTSK (0.47) CTSKCTSSALDH1A1KDM4EMAPT
SCHEMBL7303744 0.78 CTSK (0.40) CTSKCTSSKLK5KLK7CA2
SCHEMBL7314443 0.77 CTSK (0.48) CTSKCTSSKLK5
SCHEMBL7313867 0.77 CTSK (0.48) CTSKCTSSKLK5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1041064-A2 N-substituted alpha aminoacid amides as calcium channel modulators ELI LILLY AND COMPANY LIMITED (GB) 2000-10-04 EP disclosed
EP-0805147-A1 Novel N-substituted alpha aminoacid amides as calcium channel modulators LILLY INDUSTRIES LIMITED (GB) 1997-11-05 EP disclosed