SCHEMBL7305886

SCHEMBL7305886

CC(C)(C)OC(=O)C[C@H](NC(=O)CCNC(=O)Cc1ccc(C#N)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)OC(C)(C)C

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CTSS P25774 6/20 0.45
CTSB P07858 4/20 0.45
CTSL P07711 2/20 0.45
CTSK P43235 4/20 0.44
ABCB1 P08183 2/20 0.43
MAPT P10636 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
ACE P12821 1/20 0.41
KLK5 Q9Y337 1/20 0.41
MMP1 P03956 1/20 0.41
MMP3 P08254 1/20 0.41
MMP9 P14780 1/20 0.41
CCKBR P32239 1/20 0.40
PSMB8 P28062 2/20 0.40
PSMB5 P28074 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7301659 0.90 CTSG (0.46) CTSSCTSBCTSLCTSKABCB1
SCHEMBL7338218 0.88 CTSS (0.45) CTSSCTSBCTSLCTSKABCB1
SCHEMBL9215224 0.87 REN (0.48) CTSSCTSBCTSLCTSKABCB1
SCHEMBL7307169 0.86 CCKBR (0.44) CTSSCTSBCTSLMAPTTDP1
Iodide SCHEMBL9217545 0.85 CCKBR (0.42) CTSLMAPTTDP1ACEKLK5
SCHEMBL7304706 0.84 ABCB1 (0.44) CTSSCTSBCTSLCTSKABCB1
SCHEMBL9335616 0.83 LMNA (0.44) CTSLABCB1MAPTTDP1PSMB8
SCHEMBL8442775 0.82 MEN1 (0.49) CTSSCTSBCTSLCTSKABCB1
SCHEMBL9223574 0.80 CTSG (0.50) CTSSCTSBCTSLCTSKTDP1
SCHEMBL7336100 0.79 CTSL (0.49) CTSLCTSKABCB1MAPTTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0445796-B1 Derivatives of acetic acid containing peptide bonds HOFFMANN LA ROCHE (CH) 1998-06-17 EP disclosed
US-5430024-A Peptides bearing N-terminal amidino moieties and their use as inhibitors of platelet aggregation HOFFMANN-LA ROCHE INC. (US) 1995-07-04 US disclosed
US-5273982-A An amidinoaryleneamidoalkylpiperazinyleneacetic acid HOFFMANN-LA ROCHE INC. (US) 1993-12-28 US disclosed
EP-0445796-A2 Derivatives of acetic acid F. HOFFMANN-LA ROCHE AG (CH) 1991-09-11 EP disclosed