SCHEMBL7308089

SCHEMBL7308089

CCOC(=O)CCCn1c(=O)[nH]c(=O)c2ccccc21

nearest known ligand 0.62

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TNF P01375 2/20 0.62
CTNNB1 P35222 1/20 0.54
PARP1 P09874 6/20 0.53
KDM4E B2RXH2 2/20 0.51
MAPT P10636 1/20 0.48
HSD17B10 Q99714 1/20 0.48
RAB9A P51151 1/20 0.48
CNR1 P21554 1/20 0.47
GAA P10253 1/20 0.47
LMNA P02545 2/20 0.46
CREBBP Q92793 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10830938 0.85 TNF (0.58) TNFCTNNB1KDM4EMAPTHSD17B10
SCHEMBL10487972 0.85 KDM4E (0.62) CTNNB1PARP1KDM4EHSD17B10RAB9A
SCHEMBL7309296 0.84 TDP1 (0.47) TNFKDM4EHSD17B10GAALMNA
SCHEMBL7300323 0.83 HSD17B10 (0.48) TNFKDM4EMAPTHSD17B10
SCHEMBL7300140 0.82 FABP4 (0.68) CTNNB1PARP1KDM4EHSD17B10
SCHEMBL7654811 0.81 HSD17B10 (0.71) TNFKDM4EMAPTHSD17B10LMNA
SCHEMBL12938925 0.80 TNF (0.64) TNFCTNNB1KDM4ERAB9ACNR1
SCHEMBL6028786 0.80 PGR (0.60) PARP1KDM4EHSD17B10RAB9AGAA
SCHEMBL1004476 0.79 TNF (0.63) TNFCTNNB1KDM4ECNR1CREBBP
SCHEMBL1004093 0.79 TNF (0.63) TNFCTNNB1KDM4ECNR1CREBBP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5304560-A Treating CNS disorders; dopamine receptor antagonist FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1994-04-19 US disclosed
EP-0481342-A1 Quinazoline derivatives and their preparation FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1992-04-22 EP disclosed