SCHEMBL7308646

SCHEMBL7308646

CNC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)(C)c1ccccc1

nearest known ligand 0.65

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CTSS P25774 8/20 0.53
CTSL P07711 7/20 0.53
CTSB P07858 5/20 0.53
TACR1 P25103 1/20 0.51
CTSK P43235 5/20 0.50
SYK P43405 1/20 0.48
CYP3A4 P08684 3/20 0.47
CYP1A2 P05177 2/20 0.47
CYP2D6 P10635 2/20 0.47
CYP2C9 P11712 2/20 0.47
CYP2C19 P33261 2/20 0.47
ALDH1A1 P00352 2/20 0.47
TSHR P16473 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
ATM Q13315 1/20 0.47
CTRB1 P17538 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8649599 0.91 MMP2 (0.54) CTSSCTSLCTSBCTSKSYK
SCHEMBL8280590 0.91 MMP2 (0.54) CTSSCTSLCTSBCTSKSYK
SCHEMBL7307186 0.88 CTSS (0.53) CTSSCTSLCTSBTACR1CTSK
SCHEMBL29231568 0.84 CTSL (0.54) CTSSCTSLCTSBCTSKCYP3A4
SCHEMBL7761992 0.81 SYK (0.53) CTSSCTSLCTSBCTSKSYK
SCHEMBL12195056 0.79 CTSD (0.53) CTSSCTSLCTSBCTSKSYK
SCHEMBL10257423 0.79 CTSD (0.53) CTSSCTSLCTSBCTSKSYK
SCHEMBL6182844 0.79 CTSS (0.71) CTSSCTSLCTSBTACR1CTSK
SCHEMBL23604935 0.78 CTSK (0.63) CTSSCTSLCTSBCTSKCYP3A4
SCHEMBL478316 0.78 SYK (0.54) CTSSCTSLCTSBCTSKSYK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0575844-B1 Hydroxamic acid derivatives and pharmaceutical compositions thereof HOFFMANN LA ROCHE (CH) 1998-01-21 EP disclosed
EP-0575844-A2 Hydroxamic acid derivatives and pharmaceutical compositions thereof F. HOFFMANN-LA ROCHE AG (CH) 1993-12-29 EP disclosed