SCHEMBL7308820

SCHEMBL7308820

CC(C)C(C#N)(CCCNC(=O)CNCC(c1ccccc1)c1ccccc1)c1cccc(F)c1

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.38
GPR139 Q6DWJ6 2/20 0.38
ABCB1 P08183 3/20 0.37
ADRA1D P25100 1/20 0.37
ADRA1A P35348 1/20 0.37
ADRA1B P35368 1/20 0.37
OPRM1 P35372 2/20 0.36
OPRL1 P41146 2/20 0.36
CYP3A5 P20815 1/20 0.36
EBP Q15125 2/20 0.36
SIGMAR1 Q99720 2/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
TACR1 P25103 2/20 0.36
CACNA1B Q00975 2/20 0.36
POLB P06746 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7313653 0.91 EBP (0.43) CYP3A4ABCB1ADRA1DADRA1AADRA1B
SCHEMBL7311139 0.91 EBP (0.43) CYP3A4ABCB1ADRA1DADRA1AADRA1B
SCHEMBL7315211 0.90 POLB (0.39) CYP3A4ABCB1ADRA1DADRA1AADRA1B
SCHEMBL7309649 0.88 MTNR1A (0.43) CYP3A4GPR139ABCB1ADRA1AOPRM1
SCHEMBL7314600 0.84 GPR139 (0.39) CYP3A4GPR139ABCB1ADRA1DADRA1A
SCHEMBL7309023 0.83 CYP3A4 (0.42) CYP3A4ABCB1CYP3A5EBPSIGMAR1
SCHEMBL7309344 0.80 L3MBTL1 (0.37) CYP3A4ADRA1DADRA1AADRA1BL3MBTL1
SCHEMBL7313591 0.79 CCR1 (0.39) ADRA1DADRA1AADRA1BTACR1HDAC6
SCHEMBL7314922 0.75 EBP (0.43) CYP3A4ABCB1EBPSIGMAR1L3MBTL1
SCHEMBL7305541 0.74 EBP (0.43) CYP3A4ABCB1ADRA1DADRA1AADRA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1041064-A2 N-substituted alpha aminoacid amides as calcium channel modulators ELI LILLY AND COMPANY LIMITED (GB) 2000-10-04 EP disclosed
EP-0805147-A1 Novel N-substituted alpha aminoacid amides as calcium channel modulators LILLY INDUSTRIES LIMITED (GB) 1997-11-05 EP disclosed