SCHEMBL7313591

SCHEMBL7313591

CCC(C#N)(CCCNC(=O)CNCC(c1ccccc1)c1ccccc1)c1ccccc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 1/20 0.39
TACR1 P25103 4/20 0.38
CNR1 P21554 2/20 0.36
CNR2 P34972 2/20 0.36
HPGD P15428 3/20 0.35
LMNA P02545 2/20 0.35
MEN1 O00255 1/20 0.35
TP53 P04637 1/20 0.35
KMT2A Q03164 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
ADRA1D P25100 1/20 0.35
ADRA1A P35348 1/20 0.35
ADRA1B P35368 1/20 0.35
GRIN1 Q05586 2/20 0.35
GRIN2A Q12879 2/20 0.35
KDM1A O60341 1/20 0.34
HDAC3 O15379 2/20 0.34
HDAC4 P56524 2/20 0.34
HDAC1 Q13547 2/20 0.34
HDAC7 Q8WUI4 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7311139 0.83 EBP (0.43) TACR1CNR1CNR2HPGDADRA1D
SCHEMBL7313653 0.83 EBP (0.43) TACR1CNR1CNR2HPGDADRA1D
SCHEMBL7309730 0.79 CTSL (0.48)
SCHEMBL7315211 0.79 POLB (0.39) TACR1ADRA1DADRA1AADRA1B
SCHEMBL7308820 0.79 CYP3A4 (0.38) TACR1ADRA1DADRA1AADRA1BHDAC6
SCHEMBL7314600 0.77 GPR139 (0.39) CNR1CNR2ADRA1DADRA1AADRA1B
SCHEMBL7309023 0.75 CYP3A4 (0.42) CNR1CNR2HPGDMEN1KMT2A
SCHEMBL7309649 0.75 MTNR1A (0.43) MEN1KMT2AADRA1A
SCHEMBL7309344 0.74 L3MBTL1 (0.37) HPGDADRA1DADRA1AADRA1BHDAC6
SCHEMBL8016342 0.71 CCR1 (0.42) CCR1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1041064-A2 N-substituted alpha aminoacid amides as calcium channel modulators ELI LILLY AND COMPANY LIMITED (GB) 2000-10-04 EP disclosed
EP-0805147-A1 Novel N-substituted alpha aminoacid amides as calcium channel modulators LILLY INDUSTRIES LIMITED (GB) 1997-11-05 EP disclosed