SCHEMBL7315211

SCHEMBL7315211

CC(C)C(C#N)(CCCNC(=O)CNCC(c1ccccc1)c1ccccc1)c1ccc(F)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.39
EBP Q15125 2/20 0.38
SIGMAR1 Q99720 2/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
CYP3A4 P08684 3/20 0.37
ABCB1 P08183 2/20 0.37
CYP3A5 P20815 1/20 0.36
SLC6A9 P48067 3/20 0.36
ADRA1D P25100 2/20 0.36
ADRA1A P35348 2/20 0.36
ADRA1B P35368 2/20 0.36
TACR1 P25103 1/20 0.35
CACNA1B Q00975 1/20 0.35
SLC6A2 P23975 1/20 0.35
SLC6A4 P31645 1/20 0.35
SLC6A3 Q01959 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
HTT P42858 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7311139 0.93 EBP (0.43) EBPSIGMAR1L3MBTL1CYP3A4ABCB1
SCHEMBL7313653 0.93 EBP (0.43) EBPSIGMAR1L3MBTL1CYP3A4ABCB1
SCHEMBL7314600 0.90 GPR139 (0.39) EBPSIGMAR1L3MBTL1CYP3A4ABCB1
SCHEMBL7308820 0.90 CYP3A4 (0.38) POLBEBPSIGMAR1L3MBTL1CYP3A4
SCHEMBL7309023 0.89 CYP3A4 (0.42) EBPSIGMAR1CYP3A4ABCB1CYP3A5
SCHEMBL7309649 0.83 MTNR1A (0.43) CYP3A4ABCB1CYP3A5ADRA1ACACNA1B
SCHEMBL7309344 0.82 L3MBTL1 (0.37) POLBL3MBTL1CYP3A4ADRA1DADRA1A
SCHEMBL7313591 0.79 CCR1 (0.39) ADRA1DADRA1AADRA1BTACR1
SCHEMBL7314922 0.77 EBP (0.43) EBPSIGMAR1L3MBTL1CYP3A4ABCB1
SCHEMBL7316936 0.77 CTSL (0.49) CACNA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1041064-A2 N-substituted alpha aminoacid amides as calcium channel modulators ELI LILLY AND COMPANY LIMITED (GB) 2000-10-04 EP disclosed
EP-0805147-A1 Novel N-substituted alpha aminoacid amides as calcium channel modulators LILLY INDUSTRIES LIMITED (GB) 1997-11-05 EP disclosed