SCHEMBL7310868

SCHEMBL7310868

CC(C)OCCOCc1ccc(OCC(O)CN)cc1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 7/20 0.71
ADRB1 P08588 6/20 0.71
ADRB3 P13945 4/20 0.71
LMNA P02545 3/20 0.60
KMT2A Q03164 2/20 0.60
NFKB1 P19838 2/20 0.60
MEN1 O00255 1/20 0.60
THRB P10828 1/20 0.60
ALOX12 P18054 1/20 0.60
APEX1 P27695 1/20 0.60
MAPK1 P28482 1/20 0.60
SMN1; SMN2 Q16637 1/20 0.44
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
ADRA1A P35348 2/20 0.40
NR3C1 P04150 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2J2 P51589 1/20 0.40
PDE4D Q08499 1/20 0.40
TDP1 Q9NUW8 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5381741 0.86 ADRB2 (0.71) ADRB2ADRB1ADRB3LMNAKMT2A
SCHEMBL29688096 0.86 ADRB2 (0.70) ADRB2ADRB1ADRB3LMNAKMT2A
Bisoprolol SCHEMBL233810 0.83 ADRB1 (1.00) ADRB2ADRB1ADRB3LMNAKMT2A
Bisoprolol SCHEMBL20960 0.83 ADRB1 (1.00) ADRB2ADRB1ADRB3LMNAKMT2A
Bisoprolol SCHEMBL20961 0.83 ADRB1 (1.00) ADRB2ADRB1ADRB3LMNAKMT2A
Bisoprolol SCHEMBL6510329 0.83 ADRB1 (1.00) ADRB2ADRB1ADRB3LMNAKMT2A
SCHEMBL8237141 0.82 ADRB2 (0.65) ADRB2ADRB1ADRB3LMNAKMT2A
Bisoprolol SCHEMBL4269272 0.82 ADRB1 (0.98) ADRB2ADRB1ADRB3LMNAKMT2A
Bisoprolol SCHEMBL16821829 0.82 ADRB1 (0.98) ADRB2ADRB1ADRB3LMNAKMT2A
Bisoprolol SCHEMBL3137111 0.82 ADRB2 (0.98) ADRB2ADRB1ADRB3LMNAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4258062-A ISOPRENALINE ANTAGONISTS EFFECTING HEART RATE AND BLOOD PRESSURE MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1981-03-24 US disclosed
US-4171370-A Phenoxy-amino-propanols MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1979-10-16 US disclosed