SCHEMBL7311192

SCHEMBL7311192

COc1ccc(S(=O)(=O)c2c(CCC(=O)O)c(N)c(Br)c(C)c2C(=O)O)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
MEP1B Q16820 1/20 0.40
MMP2 P08253 5/20 0.39
MMP12 P39900 5/20 0.39
MMP9 P14780 4/20 0.39
FFAR1 O14842 1/20 0.39
MMP8 P22894 4/20 0.38
MMP13 P45452 4/20 0.38
MMP14 P50281 4/20 0.38
MMP16 P51512 4/20 0.38
RAPGEF4 Q8WZA2 1/20 0.38
MMP1 P03956 3/20 0.38
TP53 P04637 1/20 0.38
IMPDH2 P12268 1/20 0.38
PPARG P37231 1/20 0.37
PPARD Q03181 1/20 0.37
PPARA Q07869 1/20 0.37
KEAP1 Q14145 1/20 0.37
NFE2L2 Q16236 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7323918 0.78 TP53 (0.42) MMP2MMP12MMP9MMP8MMP13
SCHEMBL7324085 0.78 HTT (0.43) HTTNPSR1MEP1BMMP2MMP12
SCHEMBL7323700 0.76 RAPGEF4 (0.48) HTTNPSR1MMP2MMP12MMP9
SCHEMBL7317823 0.76 ALDH1A1 (0.39) MMP2MMP12MMP9MMP8MMP13
SCHEMBL7319427 0.74 RAPGEF4 (0.44) MMP2MMP12MMP9MMP8MMP13
SCHEMBL7318675 0.74 MMP2 (0.45) MMP2MMP12MMP9MMP8MMP13
SCHEMBL7311552 0.74 RAPGEF4 (0.41) HTTNPSR1MMP2MMP12MMP9
SCHEMBL7323861 0.74 MMP2 (0.41) MMP2MMP12MMP9MMP8MMP13
SCHEMBL7317729 0.73 RAPGEF4 (0.43) HTTNPSR1MMP2MMP12MMP9
SCHEMBL7323152 0.72 EGFR (0.43) NPSR1MMP2MMP12MMP9MMP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5929097-A INHIBIT TUMOR NECROSIS FACTOR-ALPHA CONVERTING ENZYME AMERICAN CYANAMID COMPANY (US) 1999-07-27 US disclosed