SCHEMBL7316541

SCHEMBL7316541

Cn1c(=O)c2c(ncn2CCN2CCC(c3ccccc3)CC2)n(C)c1=O

nearest known ligand 0.59

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.59
HTR7 P34969 1/20 0.59
HTR6 P50406 1/20 0.59
ADORA2B P29275 8/20 0.57
SMN1; SMN2 Q16637 2/20 0.57
RXFP1 Q9HBX9 2/20 0.57
HTR1A P08908 2/20 0.57
CHRM1 P11229 2/20 0.57
DRD2 P14416 2/20 0.57
ADRA1D P25100 2/20 0.57
ADRA1A P35348 2/20 0.57
ADRA1B P35368 2/20 0.57
CHRM2 P08172 1/20 0.57
TSHR P16473 1/20 0.57
MAPT P10636 1/20 0.52
LMNA P02545 1/20 0.52
KMT2A Q03164 1/20 0.52
CASP1 P29466 1/20 0.51
L3MBTL1 Q9Y468 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7320319 0.94 HTR7 (0.68) ALDH1A1HTR7HTR6ADORA2BSMN1; SMN2
SCHEMBL7313390 0.94 HTR1A (0.65) ALDH1A1HTR7HTR6ADORA2BSMN1; SMN2
SCHEMBL683615 0.91 ADORA2B (0.57) ALDH1A1HTR7HTR6ADORA2BSMN1; SMN2
SCHEMBL7306929 0.82 HTR7 (0.59) HTR7HTR6ADORA2BSMN1; SMN2RXFP1
SCHEMBL4461767 0.82 ADORA2B (0.73) ALDH1A1HTR7HTR6ADORA2BSMN1; SMN2
SCHEMBL1810048 0.82 HTR7 (0.84) ALDH1A1HTR7HTR6ADORA2BSMN1; SMN2
SCHEMBL9620744 0.81 HTR1A (0.59) ALDH1A1HTR7HTR6ADORA2BSMN1; SMN2
Tameridone SCHEMBL2109716 0.81 ADRA1D (0.51) HTR7HTR6HTR1ACHRM1DRD2
Tameridone SCHEMBL10869123 0.80 ADRA1D (0.52) HTR7HTR6HTR1ACHRM1DRD2
SCHEMBL7316547 0.80 ALDH1A1 (0.56) ALDH1A1HTR7HTR6ADORA2BSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4599337-A Antiphlogistic/antipyretic/analgesic agents containing theobromine or theophylline derivatives as active ingredient EISAI CO., LTD. (JP) 1986-07-08 US claimed
US-4599337-A Antiphlogistic/antipyretic/analgesic agents containing theobromine or theophylline derivatives as active ingredient EISAI CO., LTD. (JP) 1986-07-08 US disclosed
EP-0087810-B1 ANTIPHLOGISTIC/ANTIPYRETIC/ANALGESIC PHARMACEUTICAL COMPOSITIONS CONTAINING THEOPHYLLINE DERIVATIVES AS ACTIVE INGREDIENT Eisai Co., Ltd. (JP) 1986-06-25 EP disclosed
US-4564617-A VASODILATORS, ANALGESICS EISAI CO., LTD. (JP) 1986-01-14 US disclosed
US-4543254-A Antiphlogistic/antipyretic/analgesic agents containing theobromine or theophylline derivatives as active ingredient EISAI CO., LTD. (JP) 1985-09-24 US disclosed
US-4426383-A VASODILATION, ANALGESICS, CNS STIMULANTS, ANTIHISTAMINES EISAI CO., LTD. (JP) 1984-01-17 US disclosed