SCHEMBL7322246

SCHEMBL7322246

NC(=O)c1c(Cc2ccc(C(=O)O)cc2)ccc2ccccc12

nearest known ligand 0.50

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.50
PLA2G10 O15496 1/20 0.47
PLA2G2A P14555 1/20 0.47
NR1H4 Q96RI1 1/20 0.44
SRD5A2 P31213 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28227062 0.90 PLA2G10 (0.46) PLA2G10PLA2G2A
SCHEMBL28000844 0.83 MTNR1A (0.42) TSHR
SCHEMBL3048092 0.81 KDM4E (0.52)
SCHEMBL20370925 0.79 TSHR (0.63) TSHRNR1H4SRD5A2
SCHEMBL28918465 0.79 PLA2G2A (0.49) TSHRPLA2G10PLA2G2ANR1H4SRD5A2
SCHEMBL7786982 0.79 ROCK2 (0.50) PLA2G10PLA2G2A
SCHEMBL9517988 0.78 GPR55 (0.46)
SCHEMBL7789995 0.78 CAPN1 (0.54) PLA2G10PLA2G2A
SCHEMBL7314900 0.78 PYGL (0.43) PLA2G10PLA2G2A
SCHEMBL7313788 0.78 CAPN1 (0.48)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6251917-B1 Benzamidoaldehydes and their use as cysteine protease inhibitors BASF AKTIENGESELLSCHAFT (DE) 2001-06-26 US disclosed
US-6103720-A ENZYME INHIBITORS; ANTIICHEMIC AND -TUMOR AGENTS; STROKES; ALZEIMER'S DISEASE BASF AKTIENGESELLSCHAFT (DE) 2000-08-15 US disclosed