SCHEMBL7325665

SCHEMBL7325665

Nc1nc2ccc3nccnc3c2[nH]1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.44
KMT2A Q03164 3/20 0.44
KDM4E B2RXH2 2/20 0.44
MAPT P10636 2/20 0.44
DHFR P00374 1/20 0.44
GAA P10253 1/20 0.44
RAD52 P43351 1/20 0.44
BLM P54132 1/20 0.44
NUDT1 P36639 3/20 0.38
MEN1 O00255 2/20 0.38
MASP2 O00187 1/20 0.38
AOC3 Q16853 1/20 0.38
PLAU P00749 1/20 0.38
HTR3E A5X5Y0 1/20 0.38
HTR3B O95264 1/20 0.38
HTR3A P46098 1/20 0.38
BACE1 P56817 1/20 0.38
HTR3D Q70Z44 1/20 0.38
HTR3C Q8WXA8 1/20 0.38
ADRA2A P08913 3/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL88110 0.80 LMNA (0.50) ALDH1A1KMT2AKDM4EMAPTNUDT1
SCHEMBL29740308 0.80 LMNA (0.50) ALDH1A1KMT2AKDM4EMAPTNUDT1
SCHEMBL1490778 0.79 NUDT1 (0.42) ALDH1A1KMT2AKDM4EMAPTDHFR
SCHEMBL29740307 0.79 LMNA (0.48) ALDH1A1KMT2AKDM4EMAPTNUDT1
SCHEMBL2815837 0.77 ADRA2A (0.35) ALDH1A1KMT2AKDM4EMAPTDHFR
SCHEMBL22733525 0.77 ADRA2A (0.41) ALDH1A1KMT2AKDM4EMAPTDHFR
SCHEMBL15893398 0.77 HTR3E (0.42) ALDH1A1KMT2AKDM4EMAPTDHFR
SCHEMBL5942607 0.73 TGFBR1 (0.39) ALDH1A1KMT2AKDM4EMAPTGAA
SCHEMBL21712334 0.72 DYRK1A (0.37) ALDH1A1KMT2AKDM4EMAPTDHFR
SCHEMBL30107098 0.69 ALDH1A1 (0.42) ALDH1A1KMT2AMAPTBLMNUDT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0535104-B1 HETEROCYCLIC COMPOUNDS AND THEIR PREPARATION AND USE NOVO NORDISK AS (DK) 1996-09-04 EP disclosed
US-5276028-A Psychological disorders, anticonvulsants, anxiolytic or hypnotics and cognition activators NORDISK A/S (DK) 1994-01-04 US disclosed
EP-0535104-A1 HETEROCYCLIC COMPOUNDS AND THEIR PREPARATION AND USE. NOVO NORDISK AS (DK) 1993-04-07 EP disclosed
WO-1992000298-A1 HETEROCYCLIC COMPOUNDS AND THEIR PREPARATION AND USE NOVO NORDISK A/S (DK) 1992-01-09 WO disclosed