SCHEMBL7329284

SCHEMBL7329284

CC1CC(=O)NN=C1c1cccc(OCCNCC(O)COc2cccc3ccccc23)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 3/20 0.45
ADRB2 P07550 5/20 0.41
ADRB1 P08588 5/20 0.41
SIGMAR1 Q99720 4/20 0.41
ADRB3 P13945 4/20 0.41
HTR1A P08908 4/20 0.41
CYP1A2 P05177 3/20 0.41
CYP2D6 P10635 3/20 0.41
SLC6A4 P31645 3/20 0.41
HTR2B P41595 3/20 0.41
NR2E1 Q9Y466 3/20 0.41
ALDH1A1 P00352 3/20 0.41
HTR2A P28223 3/20 0.41
HTR2C P28335 3/20 0.41
HTR6 P50406 3/20 0.41
SMN1; SMN2 Q16637 3/20 0.41
MAPK1 P28482 3/20 0.41
SCN1A P35498 2/20 0.41
SLC10A1 Q14973 2/20 0.41
SCN2A Q99250 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7328370 0.92 HRH3 (0.47) ADRB2ADRB1SIGMAR1ADRB3HTR1A
SCHEMBL7303255 0.88 GPR119 (0.42) GPR119ADRB2ADRB1ADRB3HTR1A
SCHEMBL7303501 0.88 ADRB1 (0.49) GPR119ADRB2ADRB1ADRB3HTR1A
SCHEMBL7300352 0.85 ADRB1 (0.51) GPR119ADRB2ADRB1ADRB3HTR1A
SCHEMBL7295783 0.85 PDE3A (0.43) GPR119ADRB2ADRB1ADRB3HTR1A
SCHEMBL9687380 0.84 GPR119 (0.39) GPR119ADRB2ADRB1ADRB3HTR1A
SCHEMBL9687447 0.82 MAPK1 (0.41) GPR119ADRB2ADRB1SIGMAR1ADRB3
SCHEMBL7304449 0.81 PDE3B (0.39) GPR119ADRB2ADRB1SIGMAR1ADRB3
SCHEMBL7295549 0.80 GPR119 (0.42) GPR119
SCHEMBL7295668 0.80 GPR119 (0.42) GPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5135932-A 2-HYDROXYPROPYLAMINO-ALKYL-BENZIMIDAZOLY-5-YL DERIVATIVES AND THEIR USE IN THE TREATMENT OF HEART DISEASE DR. KARL THOMAE GMBH (DE) 1992-08-04 US disclosed
EP-0400519-A1 2-Hydroxy-n-propylamines, medicaments containing these compounds and method for preparing them Dr. Karl Thomae GmbH (DE) 1990-12-05 EP disclosed