SCHEMBL7333071

SCHEMBL7333071

N=C(NC(=O)OCc1ccccc1)c1ccc(C(=O)NCCC(=O)N[C@@H](CC(=O)OCc2ccccc2)C(=O)NCCc2ccc(OCC(=O)OCc3ccccc3)cc2)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
SMN1; SMN2 Q16637 4/20 0.42
LMNA P02545 1/20 0.42
MAPT P10636 3/20 0.42
NPC1 O15118 3/20 0.42
RAB9A P51151 3/20 0.42
CASP1 P29466 1/20 0.42
NFKB1 P19838 1/20 0.41
NFKB2 Q00653 1/20 0.41
RELA Q04206 1/20 0.41
HDAC8 Q9BY41 2/20 0.40
HDAC3 O15379 1/20 0.40
HDAC4 P56524 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC7 Q8WUI4 1/20 0.40
HDAC2 Q92769 1/20 0.40
HDAC10 Q969S8 1/20 0.40
HDAC11 Q96DB2 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9224285 0.96 CASP1 (0.47) MEN1KMT2ASMN1; SMN2LMNAMAPT
SCHEMBL9223556 0.91 SMN1; SMN2 (0.43) SMN1; SMN2NPC1RAB9AHDAC8HDAC2
SCHEMBL9223995 0.85 ITGB3 (0.46) SMN1; SMN2LMNARAB9ACASP1HDAC8
SCHEMBL7331480 0.85 ITGB3 (0.42) KMT2ASMN1; SMN2MAPTNPC1RAB9A
SCHEMBL8886008 0.83 MAPT (0.49) MEN1KMT2ASMN1; SMN2MAPTNPC1
SCHEMBL9217465 0.79 L3MBTL1 (0.43) MEN1KMT2AMAPTRAB9AHDAC8
SCHEMBL7300054 0.79 L3MBTL1 (0.43) MEN1KMT2AMAPTRAB9AHDAC8
SCHEMBL7299527 0.78 ITGB3 (0.44) MEN1KMT2ACASP1HDAC8HDAC3
SCHEMBL9221804 0.78 ITGB3 (0.44) MEN1KMT2ACASP1HDAC8HDAC3
SCHEMBL7305875 0.77 ACE (0.49) MAPTHDAC8HDAC3HDAC4HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0445796-B1 Derivatives of acetic acid containing peptide bonds HOFFMANN LA ROCHE (CH) 1998-06-17 EP disclosed
EP-0445796-A2 Derivatives of acetic acid F. HOFFMANN-LA ROCHE AG (CH) 1991-09-11 EP disclosed