SCHEMBL9223995

SCHEMBL9223995

O=C(O)NCCC(=O)N[C@@H](CC(=O)OCc1ccccc1)C(=O)NCCc1ccc(OCC(=O)OCc2ccccc2)cc1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 2/20 0.46
ITGA2B P08514 2/20 0.46
KDM4E B2RXH2 2/20 0.45
CASP1 P29466 1/20 0.45
RAB9A P51151 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
HDAC8 Q9BY41 1/20 0.44
ADAMTS5 Q9UNA0 2/20 0.43
PTPN1 P18031 1/20 0.43
TAOK1 Q7L7X3 1/20 0.43
TAOK3 Q9H2K8 1/20 0.43
ALDH1A1 P00352 1/20 0.43
EPHX2 P34913 1/20 0.42
CA5A P35218 1/20 0.42
LMNA P02545 1/20 0.42
POLB P06746 1/20 0.42
KLKB1 P03952 1/20 0.42
KLK1 P06870 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7333071 0.85 MEN1 (0.43) ITGB3ITGA2BCASP1RAB9ASMN1; SMN2
SCHEMBL7365496 0.85 ITGB3 (0.41) ITGB3ITGA2BKDM4ECASP1RAB9A
SCHEMBL9222050 0.84 PTPN1 (0.54) KDM4ERAB9ASMN1; SMN2ADAMTS5PTPN1
SCHEMBL7404441 0.83 KLK7 (0.51) CASP1HDAC8CA5A
SCHEMBL9224285 0.81 CASP1 (0.47) ITGB3ITGA2BCASP1RAB9ASMN1; SMN2
SCHEMBL9220637 0.78 CASP1 (0.55) CASP1HDAC8CA5A
SCHEMBL11709662 0.78 CA5A (0.60) CASP1SMN1; SMN2CA5A
SCHEMBL9224769 0.77 KLK7 (0.45) ITGB3ITGA2BSMN1; SMN2CA5A
SCHEMBL11714376 0.77 CTSK (0.61) RAB9ASMN1; SMN2HDAC8CA5A
SCHEMBL11707023 0.76 CA5A (0.58) CASP1SMN1; SMN2CA5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5430024-A Peptides bearing N-terminal amidino moieties and their use as inhibitors of platelet aggregation HOFFMANN-LA ROCHE INC. (US) 1995-07-04 US disclosed
US-5273982-A An amidinoaryleneamidoalkylpiperazinyleneacetic acid HOFFMANN-LA ROCHE INC. (US) 1993-12-28 US disclosed