SCHEMBL8886008

SCHEMBL8886008

COc1ccc(CCNC(=O)C(CC(=O)OCc2ccccc2)NC(=O)CNC(=O)c2ccc(-c3ccc(C(=N)NC(=O)OCc4ccccc4)cc3)cc2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.49
RAB9A P51151 2/20 0.49
POLB P06746 1/20 0.45
CTDSP1 Q9GZU7 1/20 0.45
NPC1 O15118 1/20 0.44
KMT2A Q03164 4/20 0.43
ALDH1A1 P00352 3/20 0.43
SMN1; SMN2 Q16637 3/20 0.43
MEN1 O00255 2/20 0.43
TP53 P04637 1/20 0.43
HPGD P15428 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C19 P33261 1/20 0.43
CTSS P25774 2/20 0.43
CTSK P43235 2/20 0.43
CTSL P07711 1/20 0.43
SFN P31947 1/20 0.42
GAA P10253 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7331480 0.85 ITGB3 (0.42) MAPTRAB9ANPC1KMT2AALDH1A1
SCHEMBL8408125 0.83 CTSL (0.41) MAPTKMT2AALDH1A1SMN1; SMN2CTSS
SCHEMBL9223556 0.83 SMN1; SMN2 (0.43) RAB9ANPC1SMN1; SMN2ITGB3ITGA2B
SCHEMBL7333071 0.83 MEN1 (0.43) MAPTRAB9ANPC1KMT2ASMN1; SMN2
SCHEMBL9252697 0.82 HDAC6 (0.42) MAPTKMT2ASMN1; SMN2MEN1TP53
SCHEMBL11714376 0.81 CTSK (0.61) MAPTRAB9ANPC1KMT2ASMN1; SMN2
SCHEMBL9224285 0.79 CASP1 (0.47) MAPTRAB9ANPC1KMT2ASMN1; SMN2
Hydrochloric Acid SCHEMBL8885572 0.79 ITGB3 (0.56) RAB9APOLBCTDSP1NPC1SFN
SCHEMBL9568122 0.78 CTSS (0.43) MAPTRAB9ANPC1KMT2AALDH1A1
SCHEMBL8885312 0.77 MAPT (0.55) MAPTRAB9APOLBKMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5597825-A AGGREGATION INHIBITORS DR. KARL THOMAE GMBH (DE) 1997-01-28 US disclosed
EP-0496378-B1 Biphenylderivatives, drugs containing these compounds and processes for their preparation THOMAE GMBH DR K (DE) 1995-09-20 EP disclosed
EP-0496378-A1 Biphenylderivatives, drugs containing these compounds and processes for their preparation Dr. Karl Thomae GmbH (DE) 1992-07-29 EP disclosed