SCHEMBL9224285

SCHEMBL9224285

N=C(NC(=O)OCc1ccccc1)c1ccc(C(=O)NCCC(=O)N[C@@H](CC(=O)O)C(=O)NCCc2ccc(OCC(=O)OCc3ccccc3)cc2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 6/20 0.47
ITGB3 P05106 2/20 0.44
ITGA2B P08514 2/20 0.44
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
SMN1; SMN2 Q16637 4/20 0.42
LMNA P02545 1/20 0.42
MAPT P10636 3/20 0.42
NPC1 O15118 3/20 0.42
RAB9A P51151 3/20 0.42
NFKB1 P19838 1/20 0.41
NFKB2 Q00653 1/20 0.41
RELA Q04206 1/20 0.41
FOLH1 Q04609 1/20 0.40
HDAC3 O15379 1/20 0.40
HDAC4 P56524 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC7 Q8WUI4 1/20 0.40
HDAC2 Q92769 1/20 0.40
HDAC10 Q969S8 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7333071 0.96 MEN1 (0.43) CASP1ITGB3ITGA2BMEN1KMT2A
SCHEMBL9223556 0.88 SMN1; SMN2 (0.43) ITGB3ITGA2BSMN1; SMN2NPC1RAB9A
SCHEMBL7331480 0.82 ITGB3 (0.42) ITGB3ITGA2BKMT2ASMN1; SMN2MAPT
SCHEMBL9223995 0.81 ITGB3 (0.46) CASP1ITGB3ITGA2BSMN1; SMN2LMNA
SCHEMBL7336397 0.80 ITGB3 (0.53) ITGB3ITGA2B
SCHEMBL8886008 0.79 MAPT (0.49) ITGB3ITGA2BMEN1KMT2ASMN1; SMN2
SCHEMBL9220637 0.77 CASP1 (0.55) CASP1HDAC8
SCHEMBL9217465 0.76 L3MBTL1 (0.43) ITGB3MEN1KMT2AMAPTRAB9A
SCHEMBL7300054 0.76 L3MBTL1 (0.43) ITGB3MEN1KMT2AMAPTRAB9A
SCHEMBL7306359 0.76 PRSS1 (0.46) ITGB3MEN1KMT2ASMN1; SMN2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5430024-A Peptides bearing N-terminal amidino moieties and their use as inhibitors of platelet aggregation HOFFMANN-LA ROCHE INC. (US) 1995-07-04 US disclosed
US-5273982-A An amidinoaryleneamidoalkylpiperazinyleneacetic acid HOFFMANN-LA ROCHE INC. (US) 1993-12-28 US disclosed