SCHEMBL7334046

SCHEMBL7334046

CC(C)[C@H](NC(=O)CCc1ccccn1)C(=O)N[C@@H](Cc1ccccc1)C(=O)C(F)(F)[C@H](Cc1ccccc1)NC(=O)[C@@H](NC(=O)CCc1ccccn1)C(C)C

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CA2 P00918 2/20 0.48
HTRA1 Q92743 2/20 0.44
CASP1 P29466 1/20 0.44
SMN1; SMN2 Q16637 3/20 0.44
CYP1A2 P05177 1/20 0.44
CYP2D6 P10635 1/20 0.44
MAPT P10636 1/20 0.44
TSHR P16473 1/20 0.44
KMT2A Q03164 2/20 0.43
ELANE P08246 3/20 0.42
MEN1 O00255 1/20 0.42
ALDH1A1 P00352 1/20 0.42
REN P00797 1/20 0.41
CTSD P07339 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7433505 0.83 CA2 (0.54) CA2SMN1; SMN2CYP1A2CYP2D6MAPT
SCHEMBL7269412 0.79 CA2 (0.67) CA2SMN1; SMN2CYP1A2CYP2D6MAPT
SCHEMBL6449601 0.79 CA2 (0.70) CA2SMN1; SMN2CYP1A2CYP2D6MAPT
SCHEMBL7416124 0.76 CASP3 (0.49) CA2CASP1ELANERENCTSD
SCHEMBL7415944 0.75 CASP1 (0.47) CA2CASP1SMN1; SMN2CYP1A2CYP2D6
SCHEMBL7423261 0.75 ELANE (0.47) CA2HTRA1CASP1SMN1; SMN2CYP1A2
SCHEMBL7806332 0.75 HTRA1 (0.58) HTRA1CASP1
SCHEMBL8157305 0.74 GPR132 (0.57) SMN1; SMN2CYP1A2CYP2D6MAPTTSHR
SCHEMBL9579040 0.74 CASP3 (0.46) CA2CASP1SMN1; SMN2CYP1A2CYP2D6
SCHEMBL7411626 0.73 CASP1 (0.47) CA2CASP1SMN1; SMN2CYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0997459-A1 Intermediates for preparing retroviral protease inhibiting compounds Abbott Laboratories (US) 2000-05-03 EP disclosed
US-5837873-A PROTECTED OXYDIAMINES ABBOTT LABORATORIES (US) 1998-11-17 US disclosed
US-5648497-A Retroviral protease inhibiting compounds ABBOTT LABORAOTRIES (US) 1997-07-15 US disclosed
US-5616714-A PYRIDYL, THIAZOLYL-SUBSTITUTED AMINO ACID DERIVATIVES ABBOTT LABORATORIES (US) 1997-04-01 US disclosed
US-5597926-A Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1997-01-28 US disclosed
US-5554783-A (2R, 3R, 4S, 5S)-3-ACETOXY-2,5-BIS/BENZYLOXYCARBONYLAMINO/ -4-BROMO-1,5-DIPHENYLHEXANE ABBOTT LABORATORIES (US) 1996-09-10 US disclosed
US-5541334-A TREATING HIV ABBOTT LABORATORIES (US) 1996-07-30 US disclosed
US-5354866-A Treating HIV infections ABBOTT LABORATORIES (US) 1994-10-11 US disclosed
EP-0486948-A2 Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1992-05-27 EP disclosed