SCHEMBL7336019

SCHEMBL7336019

CCOC(=O)COc1cccc(NS(=O)(=O)c2cccc3ccccc23)c1

nearest known ligand 0.54

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
BRAF P15056 1/20 0.51
PGR P06401 1/20 0.50
IDH1 O75874 1/20 0.49
ALDH1A1 P00352 2/20 0.48
HTT P42858 1/20 0.48
PFKFB3 Q16875 1/20 0.48
TSHR P16473 1/20 0.47
NPY5R Q15761 1/20 0.47
MAPT P10636 2/20 0.47
JAK2 O60674 1/20 0.47
JAK3 P52333 1/20 0.47
POLB P06746 1/20 0.46
CNR2 P34972 1/20 0.46
HDAC1 Q13547 1/20 0.45
FABP1 P07148 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7330777 0.85 PGR (0.58) BRAFPGRALDH1A1HTTPFKFB3
SCHEMBL7328941 0.84 F2 (0.55) ALDH1A1HTTMAPTSMN1; SMN2
SCHEMBL7325766 0.83 ALDH1A1 (0.58) ALDH1A1HTTMAPTPOLBFABP1
SCHEMBL7337150 0.80 ALDH1A1 (0.60) ALDH1A1HTTMAPTPOLBSMN1; SMN2
SCHEMBL7324605 0.79 ALDH1A1 (0.59) ALDH1A1POLBSMN1; SMN2
SCHEMBL7329316 0.78 LMNA (0.59) BRAFPGRALDH1A1POLBFABP1
SCHEMBL7334399 0.78 GPR119 (0.62) ALDH1A1POLBSMN1; SMN2
SCHEMBL11361752 0.77 NPY5R (0.51) ALDH1A1HTTTSHRNPY5RSMN1; SMN2
SCHEMBL9616697 0.77 PGR (0.59) BRAFPGRALDH1A1HTTPFKFB3
SCHEMBL7327897 0.76 IDH1 (0.57) BRAFIDH1ALDH1A1POLBSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0687253-B1 4-AMINOPYRIDINES, PROCESS FOR PREPARING THE SAME AND MEDICAMENTS CONTAINING THE SAME BOEHRINGER MANNHEIM GMBH (DE) 1998-12-16 EP disclosed
EP-0687253-A1 NEW 4-AMINOPYRIDINES, PROCESS FOR PREPARING THE SAME AND MEDICAMENTS CONTAINING THE SAME Roche Diagnostics GmbH (DE) 1995-12-20 EP disclosed
WO-1994020467-A1 NEW 4-AMINOPYRIDINES, PROCESS FOR PREPARING THE SAME AND MEDICAMENTS CONTAINING THE SAME BOEHRINGER MANNHEIM GMBH (DE) 1994-09-15 WO disclosed