SCHEMBL7348339

SCHEMBL7348339

CC(C)CC(C(N)=O)C(=O)N(O)c1ccc(-c2ccccc2)cc1

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GPR88 Q9GZN0 6/20 0.48
CTSS P25774 1/20 0.42
CTSK P43235 1/20 0.42
MCL1 Q07820 1/20 0.40
CTSB P07858 1/20 0.39
HPGDS O60760 1/20 0.39
ERAP2 Q6P179 1/20 0.39
ERAP1 Q9NZ08 1/20 0.39
LNPEP Q9UIQ6 1/20 0.39
PTGS2 P35354 1/20 0.38
MME P08473 1/20 0.38
ACE P12821 1/20 0.38
CPA1 P15085 1/20 0.38
ACE2 Q9BYF1 1/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29156944 0.85 RAB9A (0.42) GPR88RAB9A
SCHEMBL7358523 0.79 MMP12 (0.44) GPR88ERAP2ERAP1MMEACE
SCHEMBL7360611 0.79 ALDH1A1 (0.42) MCL1RAB9A
SCHEMBL7356404 0.78 MMP2 (0.44) NPC1RAB9ASMN1; SMN2
SCHEMBL7348766 0.76 SRC (0.41) GPR88HPGDSPTGS2
SCHEMBL2163671 0.75 GPR88 (0.46) GPR88CTSSCTSKMCL1CTSB
SCHEMBL7361196 0.74 ALOX5 (0.50) GPR88ERAP2ERAP1
SCHEMBL2163674 0.74 GPR88 (0.53) GPR88MCL1CTSB
SCHEMBL2163020 0.73 GPR88 (0.44) GPR88CTSSCTSKMCL1HPGDS
SCHEMBL2163024 0.70 GPR88 (0.56) GPR88

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1009736-A1 MALONIC ACID BASED MATRIX METALLOPROTEINASE INHIBITORS Roche Diagnostics GmbH (DE) 2000-06-21 EP disclosed
WO-1999011608-A1 MALONIC ACID BASED MATRIX METALLOPROTEINASE INHIBITORS ROCHE DIAGNOSTICS GMBH (DE) 1999-03-11 WO disclosed