SCHEMBL7350303

SCHEMBL7350303

O=S(=O)(Oc1cc(Cc2ccc(F)cc2)cc2ccoc12)C(F)(F)F

nearest known ligand 0.33

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.33
CA2 P00918 3/20 0.33
CA12 O43570 1/20 0.33
CFD P00746 1/20 0.31
DRD2 P14416 1/20 0.31
DRD4 P21917 1/20 0.31
DRD3 P35462 1/20 0.31
PTPN5 P54829 1/20 0.31
STS P08842 1/20 0.31
TRPA1 O75762 1/20 0.30
CA1 P00915 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7352238 0.90 CYP3A4 (0.36) CYP3A4CA2CA12CFDDRD2
SCHEMBL7351472 0.80 DRD2 (0.34) CYP3A4CA2DRD2DRD4DRD3
SCHEMBL7356228 0.78 TUBB4A (0.42) CYP3A4CA2TRPA1
SCHEMBL7355758 0.78 CA2 (0.41) CA2CA12DRD2DRD4DRD3
SCHEMBL7940562 0.78 CYP3A4 (0.31) CYP3A4
SCHEMBL7350220 0.78 CYP3A4 (0.31) CYP3A4
SCHEMBL2122378 0.74 PDE4A (0.35) DRD2DRD4DRD3
SCHEMBL7357481 0.72 CA6 (0.37) CA2CA1
SCHEMBL7376695 0.70 KMT2A (0.47) CYP3A4CA2CA1
SCHEMBL7354632 0.69 ALDH1A1 (0.34) CA2TRPA1CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0834508-B1 Substituted biphenyl or phenylpyridine derivatives, process for their preparation and pharmaceutical compositions containing them ADIR (FR) 2001-08-16 EP disclosed
US-5877190-A PHOSPHODIESTERASE INHIBITOR ADIR ET COMPAGNIE (FR) 1999-03-02 US disclosed
EP-0834508-A1 Substituted biphenyl or phenylpyridine derivatives, process for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1998-04-08 EP disclosed