SCHEMBL7352264

SCHEMBL7352264

COc1ccc(COc2cc(NC(C)=O)c(Cl)cc2C(=O)CCCCCl)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.52
ALDH1A1 P00352 5/20 0.52
CYP1A2 P05177 2/20 0.52
CYP2C9 P11712 2/20 0.52
CYP2C19 P33261 2/20 0.52
BRD4 O60885 3/20 0.48
MTNR1A P48039 2/20 0.44
MTNR1B P49286 2/20 0.44
LMNA P02545 3/20 0.43
POLB P06746 2/20 0.43
CYP3A4 P08684 1/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
MAPT P10636 4/20 0.42
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
HPGD P15428 2/20 0.41
AGER Q15109 1/20 0.41
GAA P10253 1/20 0.41
CHEK1 O14757 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7348962 0.92 ALDH1A1 (0.45) KDM4EALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL7359351 0.90 MGAT2 (0.47) KDM4EALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL7354465 0.90 SMN1; SMN2 (0.42) KDM4EALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL7355259 0.86 AGER (0.53) KDM4EALDH1A1LMNAPOLBRAB9A
SCHEMBL7350522 0.83 NPC1 (0.53) KDM4ELMNACYP3A4NPC1RAB9A
SCHEMBL7350242 0.82 SMN1; SMN2 (0.43) ALDH1A1LMNAMAPTKMT2AHPGD
SCHEMBL7358509 0.82 AGER (0.57) KDM4EALDH1A1LMNAPOLBRAB9A
SCHEMBL8970849 0.82 KDM4E (0.50) KDM4EALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL7360982 0.75 PGK1 (0.39) KDM4EALDH1A1LMNAPOLBNPC1
SCHEMBL8600700 0.73 KDM4E (0.47) KDM4EALDH1A1CYP1A2CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0700383-B1 NOVEL 1-PHENYLALKANONE 5-HT 4? RECEPTOR LIGANDS SYNTEX INC (US) 1998-09-23 EP disclosed
US-5763458-A NERVOUS SYSTEM DISORDERS, ANXIETY, ANTIDEPRESSANTS AND COGNITION ACTIVATORS SYNTEX (U.S.A.) INC. (US) 1998-06-09 US disclosed
WO-1994027965-A1 NOVEL 1-PHENYLALKANONE 5-HT4 RECEPTOR LIGANDS SYNTEX (U.S.A.) INC. (US) 1994-12-08 WO disclosed