SCHEMBL8970849

SCHEMBL8970849

COc1ccc(COc2cc(NC(C)=O)c(Cl)cc2CC(=O)CCCCl)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.50
ALDH1A1 P00352 3/20 0.50
CYP1A2 P05177 2/20 0.50
CYP2C9 P11712 2/20 0.50
CYP2C19 P33261 2/20 0.50
BRD4 O60885 3/20 0.46
MTNR1B P49286 3/20 0.45
MTNR1A P48039 2/20 0.45
LMNA P02545 3/20 0.44
POLB P06746 2/20 0.44
CYP3A4 P08684 1/20 0.44
MAPT P10636 4/20 0.42
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
GAA P10253 1/20 0.42
CHEK1 O14757 2/20 0.39
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA9 Q16790 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8970918 0.91 MTNR1B (0.43) KDM4EALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL8971536 0.90 MGAT2 (0.44) KDM4EALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL8971982 0.89 SMN1; SMN2 (0.41) KDM4EALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL8971117 0.85 AGER (0.47) KDM4EALDH1A1LMNAPOLBCYP3A4
SCHEMBL7352264 0.82 KDM4E (0.52) KDM4EALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL8971265 0.82 SMN1; SMN2 (0.42) ALDH1A1LMNAMAPTKMT2AGAA
SCHEMBL8970733 0.79 AGER (0.43) KDM4EALDH1A1LMNAPOLBCYP3A4
SCHEMBL8971050 0.75 PGK1 (0.39) KDM4EALDH1A1LMNAPOLBMAPT
SCHEMBL7348962 0.74 ALDH1A1 (0.45) KDM4EALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL7359351 0.72 MGAT2 (0.47) KDM4EALDH1A1CYP1A2CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0700383-A1 NOVEL 1-PHENYLALKANONE 5-HT 4? RECEPTOR LIGANDS SYNTEX (U.S.A.) INC. (US) 1996-03-13 EP disclosed