SCHEMBL8600700

SCHEMBL8600700

COc1ccc(COc2cc(NC(C)=O)c(Cl)cc2C(Cl)CCCC=O)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.47
ALDH1A1 P00352 5/20 0.47
CYP1A2 P05177 2/20 0.47
CYP2C9 P11712 2/20 0.47
CYP2C19 P33261 2/20 0.47
BRD4 O60885 4/20 0.44
LMNA P02545 3/20 0.42
POLB P06746 2/20 0.42
CYP3A4 P08684 1/20 0.42
MTNR1A P48039 2/20 0.41
MTNR1B P49286 2/20 0.41
MAPT P10636 4/20 0.39
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
GAA P10253 1/20 0.39
HPGD P15428 2/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
HDAC8 Q9BY41 1/20 0.37
ADORA3 P0DMS8 1/20 0.35
ADORA1 P30542 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8601552 0.92 KDM4E (0.39) KDM4EALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL8603828 0.90 MTNR1A (0.38) KDM4EALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL8602614 0.85 AGER (0.40) KDM4EALDH1A1LMNAPOLBMAPT
SCHEMBL7352264 0.73 KDM4E (0.52) KDM4EALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL8970849 0.72 KDM4E (0.50) KDM4EALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL8602051 0.72 MTNR1B (0.39) KDM4EALDH1A1BRD4MTNR1AMTNR1B
SCHEMBL8971582 0.69 AGER (0.45) ALDH1A1LMNAPOLBMAPTMEN1
SCHEMBL8811250 0.67 ALDH1A1 (0.43) ALDH1A1CYP1A2CYP3A4MAPTMEN1
SCHEMBL8812863 0.67 PTGER1 (0.46) CYP2C9MEN1KMT2A
SCHEMBL25267903 0.67 KDM4E (0.67) KDM4EALDH1A1CYP1A2CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5763458-A NERVOUS SYSTEM DISORDERS, ANXIETY, ANTIDEPRESSANTS AND COGNITION ACTIVATORS SYNTEX (U.S.A.) INC. (US) 1998-06-09 US disclosed