SCHEMBL7353290

SCHEMBL7353290

CC(C)(O)C[S+]([O-])c1nc2ccccc2[nH]1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DDAH1 O94760 1/20 0.41
TXN P10599 1/20 0.41
CYP1A2 P05177 2/20 0.41
CYP2C9 P11712 1/20 0.41
KDM4E B2RXH2 3/20 0.40
NPSR1 Q6W5P4 2/20 0.40
PKM P14618 2/20 0.40
ALDH1A1 P00352 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
NPC1 O15118 1/20 0.40
ABCB11 O95342 1/20 0.40
TP53 P04637 1/20 0.40
RAB9A P51151 1/20 0.40
HSD17B10 Q99714 1/20 0.40
HDAC6 Q9UBN7 1/20 0.39
MAPK1 P28482 1/20 0.39
IDO1 P14902 1/20 0.38
POLB P06746 1/20 0.38
LMNA P02545 1/20 0.38
CYP2D6 P10635 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7353284 0.85 DDAH1 (0.41) DDAH1TXNCYP1A2CYP2C9KDM4E
SCHEMBL7289169 0.80 RAB9A (0.46) DDAH1KDM4ENPSR1PKMALDH1A1
SCHEMBL9560922 0.80 DDAH1 (0.51) DDAH1TXNCYP1A2KDM4ENPSR1
SCHEMBL7288161 0.77 EPHX2 (0.46) DDAH1KDM4ENPSR1PKMALDH1A1
SCHEMBL7289165 0.76 NPC1 (0.46) DDAH1KDM4ENPSR1PKMALDH1A1
SCHEMBL11364032 0.75 CHRM1 (0.50) CYP1A2CYP2C9KDM4ENPSR1PKM
SCHEMBL7298834 0.74 L3MBTL1 (0.41) DDAH1KDM4ENPSR1PKMALDH1A1
SCHEMBL28468886 0.74 SMN1; SMN2 (0.46) DDAH1KDM4EPKMALDH1A1SMN1; SMN2
SCHEMBL2799383 0.74 ALDH1A1 (0.50) DDAH1TXNCYP1A2KDM4ENPSR1
SCHEMBL636639 0.74 GAA (0.50) DDAH1KDM4ENPSR1PKMALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5652247-A VASOPRESSIN ANTAGONIST OTSUKA PHARMACEUTICAL CO., LTD (JP) 1997-07-29 US disclosed
US-5436254-A Vaopressin antagonists OTSUKA PHARMACEUTICAL COMPANY, LTD. (JP) 1995-07-25 US disclosed
EP-0602209-A1 OXYTOCIN ANTAGONIST OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1994-06-22 EP disclosed
EP-0382185-B1 Carbostyril derivatives OTSUKA PHARMA CO LTD (JP) 1994-06-15 EP disclosed
WO-1994001113-A1 OXYTOCIN ANTAGONIST OTSUKA PHARMACEUTICAL COMPANY, LIMITED (JP) 1994-01-20 WO disclosed
US-5225402-A Vasopressin antagonist, vasodilation, hypotensive, diuretics and anticoagulants OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1993-07-06 US disclosed