SCHEMBL7360787

SCHEMBL7360787

CC(C)CCC(N)(C(=O)NC(C)(C)C)[C@H](O)[C@H](Cc1ccccc1)NC(=O)[C@H](C)NS(=O)(=O)C=Cc1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.44
POLB P06746 1/20 0.43
ADAM17 P78536 1/20 0.39
GAA P10253 1/20 0.38
ITGB3 P05106 1/20 0.34
ITGA2B P08514 1/20 0.34
BCHE P06276 1/20 0.34
PSEN1 P49768 2/20 0.34
PSEN2 P49810 2/20 0.34
APH1B Q8WW43 2/20 0.34
NCSTN Q92542 2/20 0.34
APH1A Q96BI3 2/20 0.34
PSENEN Q9NZ42 2/20 0.34
ALDH1A1 P00352 2/20 0.34
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
MAPK1 P28482 1/20 0.33
CYP2C19 P33261 1/20 0.33
EGFR P00533 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7360777 1.00 HTT (0.44) HTTPOLBADAM17GAAITGB3
SCHEMBL7424747 0.81 HTT (0.46) HTTPOLBADAM17GAABCHE
SCHEMBL7424741 0.81 HTT (0.46) HTTPOLBADAM17GAABCHE
SCHEMBL7361078 0.78 MMP2 (0.36) BCHE
SCHEMBL8882496 0.76 PSEN1 (0.38) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL7318484 0.74 LAP3 (0.49)
SCHEMBL7353045 0.74 ADAM17 (0.44) HTTPOLBADAM17GAAPSEN1
SCHEMBL7353051 0.74 ADAM17 (0.44) HTTPOLBADAM17GAAPSEN1
SCHEMBL7352170 0.73 GAA (0.39) HTTPOLBADAM17GAAITGB3
SCHEMBL7352165 0.73 GAA (0.39) HTTPOLBADAM17GAAITGB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0558673-A1 RETROVIRAL PROTEASE INHIBITORS. MONSANTO CO (US) 1993-09-08 EP disclosed
WO-1992008699-A1 RETROVIRAL PROTEASE INHIBITORS MONSANTO COMPANY (US) 1992-05-29 WO disclosed