SCHEMBL7361398

SCHEMBL7361398

COc1ccc(SCC(C(=O)O)C2(C)NC(=O)N(C)C2=O)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.37
MTNR1A P48039 1/20 0.36
MTNR1B P49286 1/20 0.36
ALDH1A1 P00352 1/20 0.36
MAPK1 P28482 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA4 P22748 1/20 0.36
CA7 P43166 1/20 0.36
CA9 Q16790 1/20 0.36
F2 P00734 1/20 0.36
LDHA P00338 1/20 0.35
MAPT P10636 1/20 0.35
PKM P14618 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
KIF11 P52732 2/20 0.35
RAB9A P51151 2/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7366561 0.79 HTT (0.42) ALDH1A1NPSR1MEN1KMT2AMMP1
SCHEMBL6379273 0.78 NPC1 (0.38) NPC1MTNR1AMTNR1BALDH1A1F2
SCHEMBL6380461 0.70 MTNR1A (0.50) NPC1MTNR1AMTNR1BALDH1A1CA1
SCHEMBL7361327 0.70 MMP1 (0.43) CA1CA2CA9MMP1MMP2
SCHEMBL12264723 0.69 MMP2 (0.49) NPC1MTNR1AMTNR1BALDH1A1CA1
SCHEMBL7075160 0.67 MTNR1A (0.47) NPC1MTNR1AMTNR1BALDH1A1CA1
SCHEMBL7074737 0.65 TAS1R3 (0.44) NPC1MTNR1AMTNR1BALDH1A1CA1
Cadaverine Tartrate SCHEMBL29661248 0.65 MTNR1A (0.51) NPC1MTNR1AMTNR1BALDH1A1CA1
SCHEMBL7073559 0.64 PDE4B (0.48) NPC1MTNR1AMTNR1BALDH1A1LDHA
SCHEMBL772862 0.64 CA1 (0.53) NPC1MTNR1AMTNR1BALDH1A1CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0929519-A1 $g(b)-SULFONYL HYDROXAMIC ACIDS AS MATRIX METALLOPROTEINASES INHIBITORS PHARMACIA & UPJOHN COMPANY (US) 1999-07-21 EP disclosed
WO-1998013340-A1 β-SULFONYL HYDROXAMIC ACIDS AS MATRIX METALLOPROTEINASES INHIBITORS PHARMACIA & UPJOHN COMPANY (US) 1998-04-02 WO disclosed