SCHEMBL7362732

SCHEMBL7362732

CC(C)n1nc(-c2c(-c3ccc(F)c(F)c3)nn3ccncc23)ccc1=O

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BMPR1B O00238 1/20 0.37
BMPR1A P36894 1/20 0.37
TGFBR1 P36897 1/20 0.37
ACVRL1 P37023 1/20 0.37
ACVR1 Q04771 1/20 0.37
CYP1A2 P05177 3/20 0.34
CYP3A4 P08684 3/20 0.34
USP2 O75604 2/20 0.34
HSD17B10 Q99714 2/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
ALDH1A1 P00352 1/20 0.34
MAPK14 Q16539 2/20 0.33
CYP11B1 P15538 1/20 0.33
CYP11B2 P19099 1/20 0.33
PGR P06401 1/20 0.33
MET P08581 1/20 0.32
HRH3 Q9Y5N1 1/20 0.32
EGFR P00533 4/20 0.32
PIK3CD O00329 3/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7362751 0.89 MAPK14 (0.42) BMPR1BBMPR1ATGFBR1ACVRL1ACVR1
SCHEMBL7366115 0.87 USP2 (0.35) BMPR1BBMPR1ATGFBR1ACVRL1ACVR1
SCHEMBL7365171 0.87 BMPR1B (0.36) BMPR1BBMPR1ATGFBR1ACVRL1ACVR1
SCHEMBL7363632 0.85 BMPR1B (0.37) BMPR1BBMPR1ATGFBR1ACVRL1ACVR1
SCHEMBL7367166 0.83 BRD4 (0.44) BMPR1BBMPR1ATGFBR1ACVRL1ACVR1
SCHEMBL7367567 0.83 MAT2A (0.33) BMPR1BBMPR1ATGFBR1ACVRL1ACVR1
SCHEMBL7366330 0.78 PDE3A (0.40) CYP1A2CYP3A4USP2HSD17B10CA1
SCHEMBL7364069 0.75 PDE1A (0.39) CYP1A2CYP3A4HSD17B10ALDH1A1MAPK14
SCHEMBL7036702 0.75 BMPR1B (0.34) BMPR1BBMPR1ATGFBR1ACVRL1ACVR1
SCHEMBL7035938 0.74 BMPR1B (0.33) BMPR1BBMPR1ATGFBR1ACVRL1ACVR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1244669-A1 PYRAZOLOPYRAZINES AND THEIR USE AS ADENOSINE ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2002-10-02 EP disclosed
WO-2001040230-A1 PYRAZOLOPYRAZINES AND THEIR USE AS ADENOSINE ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-06-07 WO disclosed