SCHEMBL7363595

SCHEMBL7363595

CC(C)Cc1nc(-c2ccncn2)oc1C(=O)C(CCNC(=O)C(C(N)=O)C1CCCCC1)c1ccccc1

nearest known ligand 0.32

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
TP53 P04637 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2D6 P10635 1/20 0.30
TSHR P16473 1/20 0.30
TDP1 Q9NUW8 1/20 0.30
REN P00797 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7364308 0.90 MEN1 (0.35) MEN1KMT2ATP53CYP1A2CYP3A4
SCHEMBL6801151 0.72 CTSL (0.39) REN
SCHEMBL6801144 0.68 CTSL (0.33) REN
SCHEMBL7363588 0.66 ALDH1A1 (0.37) TP53TSHR
SCHEMBL7365739 0.64 ERCC1 (0.36)
SCHEMBL6806942 0.61 CTSL (0.43) REN
SCHEMBL6918536 0.61 BMP1 (0.40) MEN1KMT2AREN
SCHEMBL6918534 0.61 BMP1 (0.34) REN
SCHEMBL6062675 0.61 CTSS (0.42) CYP3A4
SCHEMBL7361089 0.60 IKBKB (0.39) REN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1159273-A1 COMPOUNDS USEFUL AS REVERSIBLE INHIBITORS OF CATHEPSIN S BOEHRINGER INGELHEIM PHARMACEUTICALS INC. (US) 2001-12-05 EP disclosed
WO-2000051998-A1 COMPOUNDS USEFUL AS REVERSIBLE INHIBITORS OF CATHEPSIN S BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2000-09-08 WO disclosed