SCHEMBL7380932

SCHEMBL7380932

CC(C)(C)CC(=O)N[C@@H](Cc1ccccc1)C(=O)ONC(=O)c1cc(NC(=N)N)cc(C(F)(F)F)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RHOC P08134 1/20 0.43
RHOA P61586 1/20 0.43
NOS3 P29474 1/20 0.41
NOS1 P29475 1/20 0.41
NOS2 P35228 1/20 0.41
MDM4 O15151 1/20 0.39
MDM2 Q00987 1/20 0.39
FPR2 P25090 1/20 0.39
MEN1 O00255 1/20 0.38
ALDH1A1 P00352 1/20 0.38
LMNA P02545 1/20 0.38
KMT2A Q03164 1/20 0.38
P2RX1 P51575 1/20 0.38
MCL1 Q07820 1/20 0.38
TACR1 P25103 2/20 0.37
REN P00797 1/20 0.37
TRPA1 O75762 1/20 0.37
CYP1A2 P05177 1/20 0.37
CA12 O43570 2/20 0.37
CA1 P00915 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8428868 0.90 RHOC (0.43) RHOCRHOANOS3NOS1NOS2
SCHEMBL7375475 0.87 CA12 (0.43) MDM4MDM2ALDH1A1LMNAKMT2A
SCHEMBL7375077 0.86 RHOC (0.39) RHOCRHOANOS3NOS1NOS2
SCHEMBL7450957 0.84 ITGB1 (0.45) RHOCRHOAFPR2P2RX1TRPA1
SCHEMBL7376760 0.84 ITGB1 (0.45) RHOCRHOAFPR2P2RX1TRPA1
SCHEMBL7803127 0.82 FPR2 (0.45) RHOCRHOAFPR2P2RX1MCL1
SCHEMBL7379710 0.81 ITGB3 (0.41) RHOCRHOAP2RX1MCL1TRPA1
SCHEMBL7451739 0.79 ACE (0.45) RHOCRHOAFPR2ALDH1A1P2RX1
SCHEMBL7410384 0.75 ITGB3 (0.54) RENCA12CA1CA2CA9
SCHEMBL7380577 0.75 CTSL (0.54) ALDH1A1CA12CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0891325-A1 PARA-SUBSTITUTED PHENYLPROPANOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1999-01-20 EP claimed
WO-1997036859-A1 PARA-SUBSTITUTED PHENYLPROPANOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1997-10-09 WO claimed