SCHEMBL738536

SCHEMBL738536

O=C(c1cc(Cl)cc(Cl)c1)C(F)(F)Cl

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TPMT P51580 1/20 0.50
HCAR1 Q9BXC0 1/20 0.39
MEN1 O00255 1/20 0.37
PLA2G1B P04054 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
GAA P10253 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C19 P33261 1/20 0.37
KMT2A Q03164 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
ATG4B Q9Y4P1 1/20 0.37
RXRA P19793 2/20 0.36
RXRB P28702 2/20 0.36
TSHR P16473 1/20 0.36
RAB9A P51151 1/20 0.36
FLT1 P17948 1/20 0.34
FLT4 P35916 1/20 0.34
KDR P35968 1/20 0.34
FABP4 P15090 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL44147 0.84 TPMT (0.52) TPMTHCAR1MEN1PLA2G1BCYP1A2
SCHEMBL28482954 0.81 TPMT (0.54) TPMTHCAR1RXRARXRBTSHR
SCHEMBL19136413 0.80 TPMT (0.48) TPMTHCAR1MEN1PLA2G1BCYP1A2
SCHEMBL18536573 0.80 TPMT (0.48) TPMTHCAR1MEN1PLA2G1BCYP1A2
SCHEMBL18950065 0.80 HPGD (0.37) CYP3A4GAATSHRKDR
SCHEMBL9315494 0.79 PARP1 (0.55) GAACYP2C19RAB9APARP1
SCHEMBL10582876 0.76 SPR (0.38) TPMTMEN1CYP3A4KMT2ATSHR
SCHEMBL18950068 0.76 NOTUM (0.41) HCAR2PARP1
SCHEMBL13307210 0.76 CES2 (0.61) GAARXRARXRB
SCHEMBL18536542 0.75 TPMT (0.43) TPMTHCAR1MEN1PLA2G1BCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 33 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12595239-B2 Substituted isoxazoline derivatives BASF SE (DE) 2026-04-07 US disclosed
EP-4291551-B1 SUBSTITUTED ISOXAZOLINE DERIVATIVES BASF SE (DE) 2025-08-13 EP disclosed
US-20240140917-A1 SUBSTITUTED ISOXAZOLINE DERIVATIVES BASF SE (DE) 2024-05-02 US disclosed
EP-4291551-A1 SUBSTITUTED ISOXAZOLINE DERIVATIVES BASF SE (DE) 2023-12-20 EP disclosed
US-20230355590-A1 ISOXAZOLINE-SUBSTITUTED BENZAMIDE COMPOUND AND PESTICIDE NISSAN CHEMICAL CORPORATION (JP) 2023-11-09 US disclosed
CN-116888101-A Substituted isoxazoline derivatives 巴斯夫欧洲公司 2023-10-13 CN disclosed
WO-2022171472-A1 SUBSTITUTED ISOXAZOLINE DERIVATIVES BASF SE (DE) 2022-08-18 WO disclosed
EP-4043444-A1 SUBSTITUTED ISOXAZOLINE DERIVATIVES BASF SE (DE) 2022-08-17 EP disclosed
US-10874645-B2 Isoxazoline-substituted benzamide compound and pesticide NISSAN CHEMICAL CORPORATION (JP) 2020-12-29 US disclosed
US-20200155511-A1 ISOXAZOLINE-SUBSTITUTED BENZAMIDE COMPOUND AND PESTICIDE NISSAN CHEMICAL CORPORATION (JP) 2020-05-21 US disclosed
EP-2430089-A2 HIGH-MOLECULAR NON-POLAR BENZTRIAZOLES BASF SE (DE) 2012-03-21 EP disclosed
US-8138213-B2 Isoxazoline-substituted benzamide compound and pesticide NISSAN CHEMICAL INDUSTRIES, LTD. (JP) 2012-03-20 US disclosed
US-20110251398-A1 ISOXAZOLINE-SUBSTITUTED BENZAMIDE COMPOUND AND PESTICIDE NISSAN CHEMICAL INDUSTRIES, LTD. (JP) 2011-10-13 US disclosed
US-8022089-B2 Isoxazoline-substituted benzamide compound and pesticide NISSAN CHEMICAL INDUSTRIES, LTD. (JP) 2011-09-20 US disclosed
WO-2010130752-A2 HIGH-MOLECULAR NON-POLAR BENZTRIAZOLES BASF SE (DE) 2010-11-18 WO disclosed
US-7662972-B2 Isoxazoline-substituted benzamide compound and pesticide NISSAN CHEMICAL INDUSTRIES, LTD. (JP) 2010-02-16 US disclosed
US-20090312330-A1 ISOXAZOLINE-SUBSTITUTED BENZAMIDE COMPOUND AND PESTICIDE NISSAN CHEMICAL INDUSTRIES, LTD. (JP) 2009-12-17 US disclosed
WO-2009080427-A1 METHOD FOR PRODUCING UV-ABSORBING HYBRID MATERIALS BASF SE (DE) 2009-07-02 WO disclosed
US-20070066617-A1 Insecticidal and acaricidal activity for many agricultural insect pests, spider mites; endo- or ecto-parasiticide for mammals or birds; veterinary medicine; environmentally friendly NISSAN CHEMICAL INDUSTRIES, LTD. (JP) 2007-03-22 US disclosed
EP-1731512-A1 ISOXAZOLINE-SUBSTITUTED BENZAMIDE COMPOUND AND NOXIOUS ORGANISM CONTROL AGENT Nissan Chemical Industries, Ltd. (JP) 2006-12-13 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12595239-B2 Substituted isoxazoline derivatives CBR3, ADRA2C, CYP4Z1 TPMT 2353/4885HCAR1 1132/4885MEN1 4773/4885
US-20230355590-A1 ISOXAZOLINE-SUBSTITUTED BENZAMIDE COMPOUND AND PESTICIDE HDAC7, ACHE, BRDT TPMT 1744/4885HCAR1 3319/4885MEN1 3896/4885
US-20240140917-A1 SUBSTITUTED ISOXAZOLINE DERIVATIVES CYP4X1, PRDX5, PRDX1 TPMT 1838/4885HCAR1 3429/4885MEN1 4820/4885
US-20090312330-A1 ISOXAZOLINE-SUBSTITUTED BENZAMIDE COMPOUND AND PESTICIDE ATM, CHRM1, NAT1 TPMT 4669/4885HCAR1 3580/4885MEN1 1887/4885
US-10874645-B2 Isoxazoline-substituted benzamide compound and pesticide C3AR1, C5, C9 TPMT 4837/4885HCAR1 1014/4885MEN1 1558/4885
US-20110251398-A1 ISOXAZOLINE-SUBSTITUTED BENZAMIDE COMPOUND AND PESTICIDE CBR3, CHRM1, CBR1 TPMT 3611/4885HCAR1 219/4885MEN1 3051/4885
US-20070066617-A1 Insecticidal and acaricidal activity for many agricultural insect pests, spider mites; endo- or ecto-parasiticide for mammals or birds; veterinary medicine; environmentally friendly CHRM1, DDT, ATM TPMT 4669/4885HCAR1 3799/4885MEN1 1665/4885
US-20200155511-A1 ISOXAZOLINE-SUBSTITUTED BENZAMIDE COMPOUND AND PESTICIDE C3AR1, C5, C9 TPMT 4837/4885HCAR1 1014/4885MEN1 1558/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.