SCHEMBL7388174

SCHEMBL7388174

N=C(N)c1ccc(N2CC(CN3CCN(S(=O)(=O)c4ccc(Br)cc4OC(F)(F)F)CC3)OC2=O)cc1

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 7/20 0.42
ITGB3 P05106 8/20 0.40
ITGA2B P08514 8/20 0.40
PRSS1 P07477 7/20 0.40
PRSS2 P07478 7/20 0.40
PRSS3 P35030 7/20 0.40
F10 P00742 5/20 0.40
F2 P00734 1/20 0.39
LMNA P02545 1/20 0.38
ADRA2A P08913 2/20 0.37
NPY5R Q15761 2/20 0.37
MCHR1 Q99705 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7389682 0.89 LIPE (0.44) SIGMAR1ITGB3ITGA2BPRSS1PRSS2
SCHEMBL27515642 0.88 SIGMAR1 (0.43) SIGMAR1LMNAADRA2ANPY5RMCHR1
SCHEMBL7386030 0.85 ITGB3 (0.44) SIGMAR1ITGB3ITGA2BPRSS1PRSS2
SCHEMBL7387646 0.83 SIGMAR1 (0.51) SIGMAR1ITGB3ITGA2BPRSS1PRSS2
SCHEMBL7389131 0.82 THRB (0.42) SIGMAR1LMNAADRA2ANPY5RMCHR1
SCHEMBL7422648 0.81 ITGB3 (0.42) SIGMAR1ITGB3ITGA2BPRSS1PRSS2
SCHEMBL7387547 0.80 ITGB3 (0.44) SIGMAR1ITGB3ITGA2BPRSS1PRSS2
SCHEMBL7386899 0.80 F10 (0.46) SIGMAR1ITGB3ITGA2BPRSS1PRSS2
SCHEMBL27517334 0.80 KMT2A (0.47) SIGMAR1ITGB3ITGA2BPRSS1PRSS2
SCHEMBL7388205 0.79 ITGB3 (0.42) SIGMAR1ITGB3ITGA2BPRSS1PRSS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1056743-A1 BENZAMINE DERIVATIVES MERCK PATENT GmbH (DE) 2000-12-06 EP disclosed
WO-1999031092-A1 BENZAMINE DERIVATIVES MERCK PATENT GMBH (DE) 1999-06-24 WO disclosed