SCHEMBL7397371

SCHEMBL7397371

N=C(N)NC(C(N)=O)c1cccc(Cl)c1

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
S1PR3 Q99500 7/20 0.47
S1PR1 P21453 4/20 0.47
S1PR4 O95977 3/20 0.44
S1PR2 O95136 2/20 0.44
F10 P00742 1/20 0.43
PRSS1 P07477 1/20 0.43
SYK P43405 1/20 0.42
KEAP1 Q14145 1/20 0.42
NFE2L2 Q16236 1/20 0.42
PARP1 P09874 1/20 0.42
ADRA1D P25100 1/20 0.42
TRPM8 Q7Z2W7 1/20 0.41
MAPK1 P28482 1/20 0.40
MAPK10 P53779 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17664005 0.84 S1PR3 (0.49) S1PR3S1PR1S1PR4S1PR2SYK
SCHEMBL23716154 0.81 ROCK2 (0.48) SYKKEAP1NFE2L2PARP1ADRA1D
SCHEMBL13710935 0.81 ROCK2 (0.48) SYKKEAP1NFE2L2PARP1ADRA1D
SCHEMBL10966252 0.80 TACR3 (0.49) MAPK1
SCHEMBL13707887 0.78 ALDH1A1 (0.49) S1PR3S1PR4S1PR2SYKPARP1
SCHEMBL17664004 0.77 S1PR3 (0.54) S1PR3S1PR1S1PR4S1PR2SYK
SCHEMBL11647818 0.76 KEAP1 (0.55) S1PR3S1PR1S1PR4S1PR2KEAP1
SCHEMBL15774550 0.76 PARP1 (0.53) PARP1ADRA1DTRPM8
SCHEMBL23716111 0.74 OGG1 (0.45) SYKPARP1TRPM8
SCHEMBL5064609 0.73 PARP1 (0.50) PARP1ADRA1DTRPM8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002064211-A1 THROMBIN INHIBITORS MERCK & CO., INC. (US) 2002-08-22 WO disclosed