SCHEMBL7400518

SCHEMBL7400518

CC(CCC(=O)NCC#N)Cc1cccc(-c2ccc(-c3nn[nH]n3)cc2)c1

nearest known ligand 0.47

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CTSS P25774 16/20 0.47
CTSL P07711 13/20 0.47
CTSB P07858 10/20 0.47
CTSK P43235 6/20 0.47
CTSV O60911 8/20 0.44
XDH P47989 2/20 0.40
PTGER4 P35408 1/20 0.40
MAPT P10636 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7401952 0.82 CTSS (0.51) CTSSCTSLCTSBCTSKCTSV
SCHEMBL7400496 0.79 CTSS (0.60) CTSSCTSLCTSBCTSKCTSV
SCHEMBL7399686 0.79 CTSS (0.47) CTSSCTSLCTSBCTSKCTSV
SCHEMBL7401735 0.79 CTSS (0.48) CTSSCTSLCTSBCTSKCTSV
SCHEMBL7394745 0.77 CTSL (0.59) CTSSCTSLCTSBCTSK
SCHEMBL7392809 0.77 NTSR1 (0.45) CTSSCTSLCTSBCTSKCTSV
SCHEMBL7400028 0.77 CTSS (0.44) CTSSCTSLCTSBCTSKCTSV
SCHEMBL7395140 0.77 CTSS (0.44) CTSSCTSLCTSBCTSKCTSV
SCHEMBL7405812 0.76 CTSK (0.62) CTSSCTSLCTSBCTSK
SCHEMBL7441160 0.76 CTSS (0.43) CTSSCTSLCTSBCTSKCTSV

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001049288-A9 NOVEL COMPOUNDS AND COMPOSITIONS AS PROTEASE INHIBITORS MERCK FROSST CANADA INC (CA) 2001-10-25 WO disclosed