SCHEMBL7401472

SCHEMBL7401472

N#Cc1ccc2nc(C(CCN3C(=O)c4ccccc4C3=O)C(=O)O)[nH]c2c1

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MMP2 P08253 9/20 0.47
MMP9 P14780 9/20 0.47
PIN1 Q13526 1/20 0.46
MMP3 P08254 2/20 0.45
MMP13 P45452 2/20 0.45
NPY5R Q15761 2/20 0.40
CSNK1A1 P48729 1/20 0.39
CSNK1D P48730 1/20 0.39
GSK3B P49841 1/20 0.39
CSNK1G2 P78368 1/20 0.39
GRIN1 Q05586 1/20 0.39
GRIN2B Q13224 1/20 0.39
CFB P00751 1/20 0.39
CHEK2 O96017 1/20 0.39
ALDH1A1 P00352 1/20 0.38
POLB P06746 1/20 0.38
METAP2 P50579 1/20 0.38
METAP1 P53582 1/20 0.38
PDE10A Q9Y233 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7401476 0.74 HSD17B10 (0.45) PIN1NPY5RGRIN1GRIN2BALDH1A1
SCHEMBL7400871 0.67 TPH1 (0.43) GRIN1GRIN2BALDH1A1PDE10A
SCHEMBL14287936 0.65 SCN10A (0.56) PIN1CSNK1A1CSNK1DGSK3BCSNK1G2
SCHEMBL9314968 0.65 IDO1 (0.53) ALDH1A1POLB
SCHEMBL7406972 0.65 F2 (0.45) MMP2MMP9MMP3MMP13ALDH1A1
SCHEMBL7080833 0.65 ALDH1A1 (0.58) MMP2MMP9MMP3MMP13ALDH1A1
SCHEMBL20305429 0.64 PIN1 (1.00) PIN1CSNK1A1CSNK1DGSK3BCSNK1G2
SCHEMBL876560 0.64 SMN1; SMN2 (0.53) MMP2MMP9ALDH1A1
SCHEMBL7433448 0.64 ALDH1A1 (0.56) PIN1ALDH1A1POLB
SCHEMBL4069591 0.64 PIN1 (0.63) PIN1CSNK1A1CSNK1DGSK3BCSNK1G2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999026932-A1 BY AMIDINO GROUP SUBSTITUTED HETEROCYCLIC DERIVATIVES AND THEIR USE AS ANTICOAGULANTS AXYS PHARMACEUTICALS, INC. (US) 1999-06-03 WO disclosed