SCHEMBL7409573

SCHEMBL7409573

CC1CN(C(=O)OC(C)(C)C)[C@H]1COc1ccc(Cl)nc1

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CHRNA3 P32297 8/20 0.45
CHRNB2 P17787 9/20 0.44
CHRNA4 P43681 9/20 0.44
CHRNB4 P30926 5/20 0.44
CHRNB1 P11230 1/20 0.44
CHRNB3 Q05901 1/20 0.44
CHRNA7 P36544 1/20 0.42
GPR119 Q8TDV5 3/20 0.41
CYP2D6 P10635 3/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7409578 1.00 CHRNA3 (0.45) CHRNA3CHRNB2CHRNA4CHRNB4CHRNB1
SCHEMBL6588716 0.83 CHRNA3 (0.59) CHRNA3CHRNB2CHRNA4CHRNB4CHRNB1
SCHEMBL7472876 0.83 CHRNA3 (0.59) CHRNA3CHRNB2CHRNA4CHRNB4CHRNB1
SCHEMBL7418201 0.82 CHRNB2 (0.45) CHRNA3CHRNB2CHRNA4CHRNB4CHRNB1
SCHEMBL30079785 0.81 GPR119 (0.49) GPR119
SCHEMBL8435310 0.81 CHRNB2 (0.61) CHRNA3CHRNB2CHRNA4CHRNB4CHRNB1
SCHEMBL8437928 0.81 CHRNB2 (0.61) CHRNA3CHRNB2CHRNA4CHRNB4CHRNB1
SCHEMBL7524902 0.79 GPR119 (0.56) CHRNA3CHRNB2CHRNA4CHRNB4CHRNB1
SCHEMBL29757897 0.78 GPR119 (0.60) CHRNA3CHRNB2CHRNA4CHRNB4CHRNB1
SCHEMBL384986 0.78 GPR119 (0.60) CHRNA3CHRNB2CHRNA4CHRNB4CHRNB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1047690-A1 HETEROCYCLIC ETHER AND THIOETHER COMPOUNDS USEFUL IN CONTROLLING CHEMICAL SYNAPTIC TRANSMISSION Abbott Laboratories (US) 2000-11-02 EP disclosed
WO-1999032480-A1 HETEROCYCLIC ETHER AND THIOETHER COMPOUNDS USEFUL IN CONTROLLING CHEMICAL SYNAPTIC TRANSMISSION ABBOTT LABORATORIES (US) 1999-07-01 WO disclosed