SCHEMBL7413736

SCHEMBL7413736

CN(NC(=O)CN)c1ccc(C2(C(=O)N3CCCC3)CC2)cc1-c1ccc(C#N)cc1

nearest known ligand 0.38

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 7/20 0.38
HSD11B1 P28845 9/20 0.37
PIN1 Q13526 2/20 0.35
F2 P00734 1/20 0.34
F10 P00742 1/20 0.34
PRSS1 P07477 1/20 0.34
PRSS2 P07478 1/20 0.34
PRSS3 P35030 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7409726 0.79 CYP11B2 (0.36) KDM1APIN1
SCHEMBL7413734 0.74 HSD11B1 (0.36) KDM1AHSD11B1F2F10PRSS1
SCHEMBL5091269 0.67 HSD11B1 (0.61) HSD11B1
SCHEMBL7412573 0.67 ALDH1A1 (0.42) HSD11B1F2F10PRSS1PRSS2
SCHEMBL5089199 0.64 FASN (0.41) HSD11B1
SCHEMBL7415075 0.64 F2 (0.74) F2F10PRSS1PRSS2PRSS3
SCHEMBL8032174 0.64 F2 (0.58) HSD11B1F2F10PRSS1PRSS2
SCHEMBL5099562 0.63 NPC1 (0.43)
SCHEMBL7415072 0.62 F2 (0.48) HSD11B1F2F10PRSS1PRSS2
SCHEMBL5099064 0.61 MCHR1 (0.42) HSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6248770-B1 CARDIOVASCULAR DISORDERS BOEHRINGER INGELHEIM PHARMA KG (DE) 2001-06-19 US disclosed
EP-1095025-A2 BENZIMIDAZOLES, PRODUCTION THEREOF AND USE THEREOF AS MEDICAMENTS BOEHRINGER INGELHEIM KG (DE) 2001-05-02 EP disclosed
WO-2000001704-A2 BENZIMIDAZOLES, PRODUCTION THEREOF AND USE THEREOF AS MEDICAMENTS BOEHRINGER INGELHEIM PHARMA KG (DE) 2000-01-13 WO disclosed